Search Count: 63
![]() |
Crystal Structure Of Topoisomerase Iv From Klebsiella Pneumoniae In Complex With Dna And Bwc0977, A Dual-Targeting Broad-Spectrum Novel Bacterial Topoisomerase Inhibitor.
Organism: Klebsiella pneumoniae subsp. pneumoniae mgh 78578, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2025-11-12 Classification: ISOMERASE/DNA/ISOMERASE INHIBITOR Ligands: A1L5V |
Organism: Klebsiella pneumoniae subsp. pneumoniae mgh 78578, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: A1L5V
![]() |
Human Serf2
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2025-10-01 Classification: RNA BINDING PROTEIN |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2025-10-01
![]() |
Pcsk9 In Complex With A Cyclic Peptide Ldlr Disruptor
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2021-11-24 Classification: LIPID TRANSPORT, HYDROLASE Ligands: CA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-11-24
Ligands: CA
![]() |
Pcsk9 In Complex With Pcsk9I A 13Mer Cyclic Peptide Ldlr Disruptor
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2021-11-10 Classification: LIPID TRANSPORT, HYDROLASE Ligands: CA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: CA
![]() |
Structure Of Serratia Marcescens 2,3-Butanediol Dehydrogenase Mutant Q247A
Organism: Serratia marcescens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-12-23 Classification: OXIDOREDUCTASE Ligands: NAD, GOL, EDO, NA, ADP |
Organism: Serratia marcescens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-23
Ligands: NAD, GOL, EDO, NA, ADP
![]() |
Structure Of Serratia Marcescens 2,3-Butanediol Dehydrogenase
Organism: Serratia marcescens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-12-23 Classification: OXIDOREDUCTASE Ligands: NAD, HBR, HBS, ADP |
Organism: Serratia marcescens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-23
Ligands: NAD, HBR, HBS, ADP
![]() |
Structure Of Serratia Marcescens 2,3-Butanediol Dehydrogenase Mutant Q247A/V139Q
Organism: Serratia marcescens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2020-12-23 Classification: OXIDOREDUCTASE Ligands: NAD, NA, EDO |
Organism: Serratia marcescens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-23
Ligands: NAD, NA, EDO
![]() |
Crystal Structure Of Substrate-Free Human Neprilysin E584D.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-09-25 Classification: PEPTIDE BINDING PROTEIN Ligands: NAG, EDO, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: NAG, EDO, ZN
![]() |
Crystal Structure Of Human Neprilysin E584D In Complex With C-Type Natriuretic Peptide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-09-25 Classification: PEPTIDE BINDING PROTEIN Ligands: NAG, ZN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: NAG, ZN, CL
![]() |
High Resolution Crystal Structure Of Substrate-Free Human Neprilysin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-06-27 Classification: HYDROLASE Ligands: NAG, ZN, EDO, NO3, PEG, GOL, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-27
Ligands: NAG, ZN, EDO, NO3, PEG, GOL, PO4
![]() |
Estrogen Receptor Alpha Y537S Covalently Bound To Antagonist H3B-5942.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2018-03-21 Classification: nuclear protein/antagonist Ligands: F3D, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: F3D, EDO, DMS
![]() |
Estrogen Receptor Alpha Y537S Bound To Antagonist H3B-9224.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2018-03-21 Classification: nuclear protein/antagonist Ligands: F3D, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: F3D, EDO
![]() |
Hpad4 Crystal Complex With Bb-F-Amidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2017-05-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: SO4, CA, 8HT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: SO4, CA, 8HT
![]() |
Hpad4 Crystal Complex With Afm-30A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2017-05-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: SO4, CA, 8FQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: SO4, CA, 8FQ
![]() |
Hpad4 Crystal Complex With Afm-41A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2017-05-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: SO4, CA, 8FT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: SO4, CA, 8FT
![]() |
Hpad4 Crystal Complex With Afm-14A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-05-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: SO4, CA, 8FW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: SO4, CA, 8FW
![]() |
Crystal Structure Of Fgfr1-Y563C (Fgfr4 Surrogate) Covalently Bound To H3B-6527
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-05-24 Classification: transferase/transferase inhibitor Ligands: 9ES, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 9ES, SO4, EDO
![]() |
Mek1 Adopts Dfg-Out Conformation When Bound To An Analog Of E6201.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-05-03 Classification: Transferase/Transferase Inhibitor Ligands: E62, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-03
Ligands: E62, MG
![]() |
Human Angiogenin Pd Variant H13R
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-02-22 Classification: HYDROLASE Ligands: TAR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: TAR
![]() |
Human Angiogenin Als Variant K40R
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2017-02-22 Classification: HYDROLASE Ligands: TAR, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: TAR, PEG
