Search Count: 3
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Discovery And Clinical Validation Of Rly-4008, The First Highly Selective Fgfr2 Inhibitor With Activity Across Fgfr2 Alterations And Resistance Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.79 Å Release Date: 2023-06-07 Classification: TRANSFERASE/INHIBITOR Ligands: WCJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: WCJ
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Structure Of Ret Protein Tyrosine Kinase In Complex With Pralsetinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-11-11 Classification: Transferase/Transferase inhibitor Ligands: Q4J, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-11
Ligands: Q4J, FMT
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Structure Of Ret Protein Tyrosine Kinase In Complex With Selpercatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2020-11-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Q6G, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-11
Ligands: Q6G, FMT
