Search Count: 44
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Erap1 In Complex With (3S,4S)-1-(3-Cyano-6-Methylpyridin-2-Yl)-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2026-07-08 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: ZN, PO4, EDO, A1JVC
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Erap1 In Complex With (3R,4R)-1-(3-Cyano-6-Methylpyridin-2-Yl)-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2026-07-08 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: ZN, PO4, EDO, A1JVB
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Erap1 In Complex With (3R,4R)-1-[3-Cyano-6-(Cyclopropylamino)Pyridin-2-Yl]-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2026-07-08 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: ZN, PO4, EDO, A1JVL
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Erap1 In Complex With (3R,4R)-1-{3-Cyano-4-Methyl-6-[(4-Methyloxan-4-Yl)Amino]Pyridin-2-Yl}-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2026-07-08 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JV2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: ZN, PO4, EDO, A1JV2
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Erap1 In Complex With 1-[2-(5-Bromo-7-Fluoro-2-Oxo-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]-4,4-Difluorocyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2026-05-06 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, SIN, PO4, EDO, A1JVE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-06
Ligands: ZN, SIN, PO4, EDO, A1JVE
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Erap1 In Complex With 1-[2-(6-Bromo-2,2-Difluoro-3-Oxo-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2026-04-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-22
Ligands: ZN, PO4, EDO, A1JVD
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Erap1 In Complex With 1-[2-(2-Oxo-5-Phenyl-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2026-04-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, MLT, EDO, A1JVG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-22
Ligands: ZN, MLT, EDO, A1JVG
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Erap1 In Complex With 1-[2-(5-Chloro-2-Oxo-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2026-04-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-22
Ligands: ZN, PO4, EDO, A1JVH
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Erap1 In Complex With 1-[2-(3-Oxo-6-Phenyl-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2026-04-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1JVF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-22
Ligands: ZN, PO4, EDO, A1JVF
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Erap1 In Complex With 1-[2-(3-Oxo-3,4-Dihydro-2H-1,4-Benzothiazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2025-01-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, B3P, EDO, BR, A1IMK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: ZN, B3P, EDO, BR, A1IMK
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Erap1 In Complex With 1-[2-(6-Bromo-3-Oxo-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]-4,4-Difluorocyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2025-01-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1IMJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: ZN, PO4, EDO, A1IMJ
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Erap1 In Complex With 1-[2-(6-Chloro-3-Oxo-3,4-Dihydro-2H-1,4-Benzothiazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2025-01-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, MLT, EDO, A1IMM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: ZN, MLT, EDO, A1IMM
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Erap1 In Complex With 1-[2-(2-Oxo-5-Phenyl-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2025-01-22 Classification: PEPTIDE BINDING PROTEIN Ligands: ZN, PO4, EDO, A1IML |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: ZN, PO4, EDO, A1IML
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Crystal Structure Of The Open Conformation Of Insulin-Regulated Aminopeptidase In Complex With A Small-Mw Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2024-09-04 Classification: HYDROLASE Ligands: NAG, WC3, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: NAG, WC3, ZN
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Insulin Regulated Aminopeptidase (Irap) In Complex With An Allosteric Aryl Sulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2024-01-31 Classification: HYDROLASE Ligands: NAG, MLT, ZN, UKG, PEG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-31
Ligands: NAG, MLT, ZN, UKG, PEG, EDO
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Insulin-Regulated Aminopeptidase (Irap) In Complex With An Allosteric Benzopyran-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.03 Å Release Date: 2024-01-31 Classification: HYDROLASE Ligands: ZN, UJX, NAG, PEG, EDO, GLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-31
Ligands: ZN, UJX, NAG, PEG, EDO, GLY
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High-Resolution Crystal Structure Of Erap1 With Bound Bestatin Analogue Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2022-07-27 Classification: HYDROLASE Ligands: NAG, ZN, I88, EDO, MLT, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-27
Ligands: NAG, ZN, I88, EDO, MLT, PGE
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Crystal Structure Of Endoplasmic Reticulum Aminopeptidase 2 (Erap2) Complex With A Highly Selective And Potent Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2022-07-20 Classification: IMMUNE SYSTEM,HYDROLASE/INHIBITOR Ligands: ZN, GIY, EPE, MES, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: ZN, GIY, EPE, MES, NA
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Insulin Regulated Aminopeptidase (Irap) In Complex With A Nanomolar Alpha Hydroxy Beta Amino Acid Based Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2022-07-20 Classification: HYDROLASE Ligands: ZN, NAG, KFR, EDO, PEG, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: ZN, NAG, KFR, EDO, PEG, TRS
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Endoplasmic Reticulum Aminopeptidase 2 Complexed With A Hydroxamic Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2022-06-22 Classification: HYDROLASE Ligands: ZN, NAG, P4G, UQE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-22
Ligands: ZN, NAG, P4G, UQE, EDO
