Search Count: 72
![]() |
Human Jnk2 Bound To Covalent Inhibitor Yl2056
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2023-06-28 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: Y56 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-28
Ligands: Y56
![]() |
Crystal Structure Of Amp-Bound Human Jnk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2022-06-22 Classification: TRANSFERASE Ligands: AMP, P6G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-22
Ligands: AMP, P6G
![]() |
Structural Basis Of Impaired Hydrolysis In Kras Q61H Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2020-04-15 Classification: HYDROLASE Ligands: GTP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: GTP, MG
![]() |
Hras G12S In Complex With Gdp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-04-15 Classification: HYDROLASE Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: GDP, MG
![]() |
Gdp-Bound Kras P34R Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2020-04-15 Classification: HYDROLASE Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: GDP, MG
![]() |
Kras P34R Mutant Structure In Complex With Gtp Analogue
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-04-15 Classification: HYDROLASE Ligands: GNP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: GNP, MG
![]() |
Crystal Structure Of Human Kras P34R Mutant In Complex With Gnp And Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-03-11 Classification: HYDROLASE Ligands: GNP, MG, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-11
Ligands: GNP, MG, PO4
![]() |
Crystal Structure Of Human Kras P34R Mutant In Complex With Gnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-02-26 Classification: HYDROLASE Ligands: MG, PO4, GNP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: MG, PO4, GNP
![]() |
Dgy-06-116, A Novel And Selective Covalent Inhibitor Of Src Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2019-07-31 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HVY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: HVY
![]() |
Crystal Structure Of Kras V14I-Gdp Demonstrating Open Switch 1 Conformation - Form 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-07-31 Classification: HYDROLASE Ligands: GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: GDP
![]() |
Crystal Structure Of Kras V14I-Gdp Demonstrating Disorder Switch 1 Conformation - Form 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-07-31 Classification: HYDROLASE Ligands: GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: GDP
![]() |
Crystal Structure Of Kras A146T-Gdp Demonstrating Open Switch 1 Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2019-05-22 Classification: HYDROLASE Ligands: GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: GDP
![]() |
Src Kinase Bound To Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-02-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6H3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: 6H3
![]() |
Crystal Structure Of Erk2 Covalently Bound To Sm1-71
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: SO4, 6H3, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: SO4, 6H3, EDO, CL
![]() |
Crystal Structure Of Erk1 Covalently Bound To Sm1-71
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: 6H3, EWH, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: 6H3, EWH, SO4, EDO
![]() |
Kras Mutant-D33E In Gdp-Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2018-01-24 Classification: HYDROLASE Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-24
Ligands: GDP, MG
![]() |
Kras Mutant-A59G In Gdp-Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-01-24 Classification: HYDROLASE Ligands: MG, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-24
Ligands: MG, GDP
![]() |
Crystal Structure Of Human Kras A59G Mutant In Complex With Gcp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-01-24 Classification: HYDROLASE Ligands: GCP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-24
Ligands: GCP
![]() |
Crystal Structure Of Takinib Bound To Tak1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2017-08-30 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: EDH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-30
Ligands: EDH
![]() |
Kras G12C In Bound To Quinazoline Based Switch Ii Pocket (Swiip) Binder
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2017-08-23 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: GDP, MG, 8ZG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-23
Ligands: GDP, MG, 8ZG
