Search Count: 20
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Bace-1 In Complex With Compound #6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2021-07-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZQS, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-21
Ligands: ZQS, GOL
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Bace-1 In Complex With Compound #22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2021-07-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZR7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-21
Ligands: ZR7, SO4
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Bace-1 In Complex With Compound #18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2021-07-14 Classification: HYDROLASE Ligands: ZRD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ZRD, GOL, SO4
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Ror Gamma In Complex With Scr2 And Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2021-04-21 Classification: SIGNALING PROTEIN Ligands: WB7, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: WB7, GOL
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Bace-1 In Complex With Compound #3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2019-12-11 Classification: HYDROLASE/INHIBITOR Ligands: QJJ, QJM, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: QJJ, QJM, GOL, SO4
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Bace-1 In Complex With Compound #17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2019-12-11 Classification: HYDROLASE/INHIBITOR Ligands: QJV, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: QJV, GOL, SO4
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Bace-1 In Complex With Compound #18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2019-12-11 Classification: HYDROLASE/INHIBITOR Ligands: QJP, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: QJP, GOL, SO4
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Bace-1 In Complex With Compound #32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2019-12-11 Classification: HYDROLASE/INHIBITOR Ligands: QKA, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: QKA, GOL, SO4
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Bace-1 In Complex With Compound #34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2019-12-11 Classification: HYDROLASE/INHIBITOR Ligands: QK7, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: QK7, GOL, SO4
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Crystal Structure Of The Rar Alpha Ligand-Binding Domain In Complex With An Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-06-22 Classification: TRANSCRIPTION Ligands: 6Q7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 6Q7
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Bace Crystal Structure With Bicyclic Aminothiazine Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2015-06-10 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 4RW, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: 4RW, GOL
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Bace Crystal Structure With Bicyclic Aminothiazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2015-06-10 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 4RZ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: 4RZ, GOL
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Bace Crystal Structure With Tricyclic Aminothiazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-06-10 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 4RX, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: 4RX, GOL
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Bace Crystal Structure With Tricyclic Aminothiazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2015-06-10 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 4RY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: 4RY
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Crystal Structure Of Bace With Amino Thiazine Inhibitor Ly2811376
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2015-04-01 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 4B2, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-01
Ligands: 4B2, GOL
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Crystal Structure Of Bace With Amino Thiazine Inhibitor Ly2886721
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2014-12-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 3YS, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3YS, GOL
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Crystal Structure Of Human Adamts-4 In Complex With Inhibitor (Compound 1, 2-(4-Chlorophenoxy)-N-{[(4R)-4-Methyl-2,5-Dioxoimidazolidin-4-Yl]Methyl} Acetamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2014-12-10 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA, 3PQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: ZN, CA, 3PQ
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Crystal Structure Of Human Adamts-4 In Complex With Inhibitor 5-Chloro-N-{[(4R)-2,5-Dioxo-4-(1,3-Thiazol-2-Yl)Imidazolidin-4-Yl]Methyl}-1-Benzofuran-2-Carboxamide (Compound 10)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2014-12-10 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA, EDO, 3PU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: ZN, CA, EDO, 3PU
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Crystal Structure Of Human Adamts-4 In Complex With Inhibitor 5-Chloro-N-{[(4S)-4-(1-Methyl-1H-Imidazol-2-Yl)-2,5-Dioxoimidazolidin-4-Yl]Methyl}-1-Benzofuran-2-Carboxamide (Compound 11)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-12-10 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA, EDO, 3PW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: ZN, CA, EDO, 3PW
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Crystal Structure Of C-Met In Complex With Ly2801653
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-04-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: L1X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-10
Ligands: L1X
