Search Count: 10
![]() |
Inhibition Of Human Menin By Sndx-5613
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2022-12-14 Classification: TRANSCRIPTION Ligands: OQ4, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-14
Ligands: OQ4, MG
![]() |
Inhibition Of Human Menin By Sndx-5613
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2022-12-14 Classification: TRANSCRIPTION Ligands: OQ4, EDO, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-14
Ligands: OQ4, EDO, MES
![]() |
Crystal Structure Of Brd9 Bromodomain In Complex With Compound Ea-89
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2022-08-10 Classification: TRANSCRIPTION Ligands: L8L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: L8L
![]() |
Glycogen Synthase Kinase 3 Beta Complexed With Brd0209
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VK
![]() |
Glycogen Synthase Kinase 3 Beta Complexed With Brd0705
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VL
![]() |
Glycogen Synthase Kinase 3 Beta Complexed With Brd3731
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VM
![]() |
Exploiting An Asp-Glu Switch In Glycogen Synthase Kinase 3 To Design Paralog Selective Inhibitors For Use In Acute Myeloid Leukemia
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: 6VL
![]() |
Solution Structure Of The N-Terminal Dimerisation Domain Of Sgt2
Organism: Saccharomyces cerevisiae
Method: SOLUTION NMR Release Date: 2013-01-16 Classification: CHAPERONE |
Organism: Saccharomyces cerevisiae
Method: SOLUTION NMR
Release Date: 2013-01-16
![]() |
Structure Of The Complex Between The N-Terminal Dimerisation Domain Of Sgt2 And The Ubl Domain Of Get5
Organism: Saccharomyces cerevisiae
Method: SOLUTION NMR Release Date: 2013-01-16 Classification: CHAPERONE |
Organism: Saccharomyces cerevisiae
Method: SOLUTION NMR
Release Date: 2013-01-16
![]() |
Crystal Structure Of The Ubl Domain Of Mdy2 (Get5) At 1.78A
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2012-11-14 Classification: PROTEIN BINDING Ligands: SO4 |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: SO4
