Search Count: 10
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Crystal Structure Of Nlrp3 In Complex With Inhibitor Np3-742
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2025-10-22 Classification: IMMUNE SYSTEM Ligands: A1JNK, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-22
Ligands: A1JNK, ADP
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Il-1Beta In Complex With Macrocyclic Peptide Hit
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-05-22 Classification: CYTOKINE |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2024-05-22
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Il-1Beta In Complex With Covalent Del Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2024-05-22 Classification: CYTOKINE Ligands: A1H4A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-22
Ligands: A1H4A
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Human Il-1Beta, Unliganded
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2024-03-06 Classification: CYTOKINE Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-06
Ligands: SO4
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Apo Structure Of Wt Lipoprotein Lipase In Complex With Gpihbp1 Mutant N78D N82D Produced In Gnti-Deficient Hek293-F Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2019-05-08 Classification: HYDROLASE/PROTEIN BINDING Ligands: NAG, MLI, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: NAG, MLI, CA
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Apo Structure Of Wt Lipoprotein Lipase In Complex With Gpihbp1 Mutant N78D N82D Produced In Hek293-F Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.04 Å Release Date: 2019-05-08 Classification: HYDROLASE/PROTEIN BINDING Ligands: NAG, EDO, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: NAG, EDO, CA
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Compound 2 Bound Structure Of Wt Lipoprotein Lipase In Complex With Gpihbp1 Mutant N78D N82D Produced In Hek293-F Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2019-05-08 Classification: HYDROLASE/PROTEIN BINDING Ligands: NAG, M3D, EDO, CA, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: NAG, M3D, EDO, CA, TRS
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Discovery Of Imidazoquinolines As A Novel Class Of Potent, Selective And In Vivo Efficacious Cot Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-08-24 Classification: TRANSFERASE Ligands: 6DA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-24
Ligands: 6DA
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Crystal Structure Of Cot Kinase Domain In Complex With 5-(2-Amino-5-(Quinolin-3-Yl)Pyridin-3-Yl)-1,3,4-Oxadiazole-2(3H)-Thione
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2015-05-06 Classification: TRANSFERASE Ligands: 49B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 49B
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Crystal Structure Of Cot Kinase Domain In Complex With 5-(5-(1H-Indol-3-Yl)-1H-Pyrrolo[2,3-B]Pyridin-3-Yl)-1,3,4-Oxadiazol-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2015-05-06 Classification: TRANSFERASE Ligands: 499 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 499
