Search Count: 29
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Gsk-3Beta With Inhibitor 6-Chloro-N-Cyclohexyl-4-(1H-Pyrrolo[2,3-B]Pyridin-3-Yl)Pyridin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.12 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: IQ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: IQ6
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Egfr Kinase Domain Complexed With An Imidazo[2,1-B]Thiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-03-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ITI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-02
Ligands: ITI
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Ligand Bound To A Model Peptide That Mimics The Open Fusogenic Form
Organism: Escherichia coli
Method: SOLUTION NMR Release Date: 2010-01-19 Classification: UNKNOWN FUNCTION Ligands: XIG |
Organism: Escherichia coli
Method: SOLUTION NMR
Release Date: 2010-01-19
Ligands: XIG
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Discovery Of 3H-Benzo[4,5]Thieno[3,2-D]Pyrimidin-4-Ones As Potent, Highly Selective And Orally Bioavailable Pim Kinases Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: LXG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: LXG
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Discovery Of 3H-Benzo[4,5]Thieno[3,2-D]Pyrimidin-4-Ones As Potent, Highly Selective And Orally Bioavailable Pim Kinases Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: LYG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: LYG
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Discovery Of 3H-Benzo[4,5]Thieno[3,2-D]Pyrimidin-4-Ones As Potent, Highly Selective And Orally Bioavailable Pim Kinases Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: LWG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: LWG
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Structure Of H-Chk1 Complexed With A767085
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: 76A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: 76A
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Structure Of H-Chk1 Complexed With Aa582939
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: A58 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: A58
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Structure Of H-Chk1 Complexed With A771129
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: 77A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: 77A
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Structure Of H-Chk1 Complexed With A780125
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: A25 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: A25
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Structure Of H-Chk1 Complexed With A859017
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: 85A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: 85A
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Crystal Structure Of Human Dipeptidyl Peptidase Iv (Dpp Iv) Complexed With Abt-341, A Cyclohexene-Constrained Phenethylamine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-10-09 Classification: HYDROLASE Ligands: KIQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-10-09
Ligands: KIQ
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Human Dipeptidyl Peptidase Iv (Dpp4) With Piperidine-Constrained Phenethylamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2007-04-24 Classification: HYDROLASE Ligands: MA9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-04-24
Ligands: MA9
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Human Dipeptidyl Peptidase Iv (Dpp4) With Piperidinone-Constrained Phenethylamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2007-04-03 Classification: HYDROLASE Ligands: GGO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-04-03
Ligands: GGO
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Crystal Structure Of Human Dipeptidyl Peptidase 4 (Dpp Iv) With Potent Alkynyl Cyanopyrrolidine (Abt-279)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2006-12-12 Classification: HYDROLASE Ligands: AXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-12-12
Ligands: AXD
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Rat Dpp-Iv With Xanthine Mimetic Inhibitor #7
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2006-12-12 Classification: HYDROLASE Ligands: LIR |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2006-12-12
Ligands: LIR
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Native Dpp-Iv (Cd26) From Rat
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2006-07-04 Classification: HYDROLASE Ligands: NAG |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2006-07-04
Ligands: NAG
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Rat Dpp-Iv With Alkynyl Cyanopyrrolidine #1
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2006-07-04 Classification: HYDROLASE Ligands: AIA |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2006-07-04
Ligands: AIA
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Rat Dpp-Iv With Alkynyl Cyanopyrrolidine #2
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2006-07-04 Classification: HYDROLASE Ligands: SO4, 1AD |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2006-07-04
Ligands: SO4, 1AD
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Rat Dpp-Iv With Xanthine Inhibitor 4
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2006-07-04 Classification: HYDROLASE Ligands: XIH |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2006-07-04
Ligands: XIH
