Search Count: 21
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Crystal Structure Of Gsk6157 Bound To Perk (R587-R1092, Delete A660-T867) At 2.34A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2014-09-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 27D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 27D
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Crystal Structure Of Gsk6414 Bound To Perk (R587-R1092, Delete A660-T867) At 2.28 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 0WH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: GOL, 0WH
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Crystal Structure Of Gsk6924 Bound To Perk (R587-R1092, Delete A660-T867) At 2.70 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 924 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: 924
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X-Ray Crystal Structure Of A Potent Liver X Receptor Modulator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2010-04-07 Classification: TRANSCRIPTION Ligands: G58 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-04-07
Ligands: G58
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The Wild Type Androgen Receptor Ligand Binding Domain Bound With Testosterone And An Ar 20-30 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2007-07-24 Classification: HORMONE Ligands: SO4, TES, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-07-24
Ligands: SO4, TES, GOL
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The Wild Type Androgen Receptor Ligand Binding Domain Bound With Testosterone And A Tif2 Box 3 Coactivator Peptide 740-753
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2007-07-24 Classification: HORMONE Ligands: SO4, TES, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-07-24
Ligands: SO4, TES, GOL
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The Androgen Receptor Prostate Cancer Mutant H874Y Ligand Binding Domain Bound With Testosterone And An Ar 20-30 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2007-07-24 Classification: HORMONE Ligands: SO4, TES, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-07-24
Ligands: SO4, TES, GOL
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The Androgen Receptor Prostate Cancer Mutant H874Y Ligand Binding Domain Bound With Testosterone And A Tif2 Box3 Coactivator Peptide 740-753
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2007-07-24 Classification: HORMONE Ligands: TES, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-07-24
Ligands: TES, GOL
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Progesterone Receptor With Bound Asoprisnil And A Peptide From The Co-Repressor Smrt
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-03-20 Classification: TRANSCRIPTION Ligands: AS0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
Ligands: AS0
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Progesterone Receptor With Bound Asoprisnil And A Peptide From The Co-Repressor Ncor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2007-03-20 Classification: TRANSCRIPTION Ligands: AS0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
Ligands: AS0
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Crystal Structure Of The Human Androgen Receptor Ligand Binding Domain Bound With Tif2(Iii) 740-753 Peptide And R1881
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2005-08-30 Classification: TRANSCRIPTION Ligands: R18 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-08-30
Ligands: R18
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Mineralocorticoid Receptor With Bound Aldosterone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2005-07-26 Classification: TRANSCRIPTION Ligands: BOG, SO4, AS4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-07-26
Ligands: BOG, SO4, AS4, GOL
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Mineralocorticoid Receptor With Bound Progesterone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2005-07-26 Classification: TRANSCRIPTION Ligands: STR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-07-26
Ligands: STR
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Mineralocorticoid Receptor S810L Mutant With Bound Progesterone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2005-07-26 Classification: TRANSCRIPTION Ligands: STR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-07-26
Ligands: STR
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Mineralocorticoid Receptor With Bound Deoxycorticosterone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2005-07-26 Classification: TRANSCRIPTION Ligands: SO4, 1CA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-07-26
Ligands: SO4, 1CA, GOL
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Mineralocorticoid Receptor Double Mutant With Bound Cortisone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2005-07-26 Classification: TRANSCRIPTION Ligands: SO4, PDN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-07-26
Ligands: SO4, PDN
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Mineralocorticoid Receptor Double Mutant With Bound Spironolactone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2005-07-26 Classification: TRANSCRIPTION Ligands: SNL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-07-26
Ligands: SNL, SO4
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Crystal Structure Of The Human Androgen Receptor Ligand Binding Domain Bound With An Androgen Receptor Nh2-Terminal Peptide, Ar20-30, And R1881
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2004-11-16 Classification: TRANSCRIPTION Ligands: R18 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-11-16
Ligands: R18
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Crystal Structure Of The Human Androgen Receptor Ligand Binding Domain Bound With R1881
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2004-11-16 Classification: TRANSCRIPTION Ligands: R18 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-11-16
Ligands: R18
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Crystal Structure Of A Dimer Complex Of The Human Glucocorticoid Receptor Ligand-Binding Domain Bound To Dexamethasone And A Tif2 Coactivator Motif
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2003-07-15 Classification: HORMONE/HORMONE ACTIVATOR Ligands: BOG, DEX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-07-15
Ligands: BOG, DEX
