Search Count: 24
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Cryoem Structure Of Nlrp3 Nacht Domain In Complex With G2394
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2022-11-02 Classification: HYDROLASE Ligands: MG, ADP, WTN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2022-11-02
Ligands: MG, ADP, WTN
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Crystal Structure Of Lysine Specific Demethylase 1 (Lsd1) With Cc-90011
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2020-10-21 Classification: FLAVOPROTEIN Ligands: V0Y, FAD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-21
Ligands: V0Y, FAD
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Crystal Structure Of Brd4 With Qc4956
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2018-05-02 Classification: GENE REGULATION/INHIBITOR Ligands: F5V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: F5V
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Crystal Structure Of Brd4 With Qc4956
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2018-05-02 Classification: GENE REGULATION/INHIBITOR Ligands: F5Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: F5Y
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Crystal Structure Of Kdm4A With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2018-04-18 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, QC1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-18
Ligands: NI, ZN, QC1
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Crystal Structure Of Kdm4A With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2018-04-18 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, QC2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-18
Ligands: NI, ZN, QC2
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Crystal Structure Of Kdm4 With The Small Molecule Inhibitor Qc6352
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2017-09-27 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, 9DJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: NI, ZN, 9DJ
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Crystal Structure Of Human Kdm4 With Small Molecule Inhibitor Qc5714
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2017-09-27 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, 9FJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: NI, ZN, 9FJ
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Crystal Structure Of Plk1 In Complex With A Novel 5,6-Dihydroimidazolo[1,5-F]Pteridine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-02-22 Classification: Transferase/Transferase Inhibitor Ligands: 79D, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 79D, ZN
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Crystal Structure Of Plk1 In Complex With A Novel 5,6-Dihydroimidazolo[1,5-F]Pteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-02-22 Classification: Transferase/Transferase Inhibitor Ligands: ZN, 79C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: ZN, 79C
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Crystal Structure Of Plk1 In Complex With A Pyrimidodiazepinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J3, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: 1J3, ZN, ACT
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Crystal Structure Of Plk1 In Complex With Tak-960
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, ACT, 1J4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: ZN, ACT, 1J4
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Crystal Structure Of Human Dipeptidyl Peptidase Iv In Complex With A Pyridopyrimidinedione Analogue
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-02-27 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0WG, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-27
Ligands: 0WG, NAG
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With Tak-322
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, T22 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: NAG, T22
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With A Pyrimidinedione Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: RUF, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: RUF, NAG
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With A Pyrimidinedione Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: XIH, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: XIH, NAG
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With A Pyrimidinone Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: RUM, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: RUM, NAG
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Post-Insertion Complex Of The Y-Family Dna Polymerase Dpo4 With M1Dg Containing Template Dna
Organism: Sulfolobus solfataricus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-06-16 Classification: TRANSFERASE Ligands: DGT, CA |
Organism: Sulfolobus solfataricus
Method: X-RAY DIFFRACTION
Release Date: 2009-06-16
Ligands: DGT, CA
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Non-Productive Complex Of The Y-Family Dna Polymerase Dpo4 With Dgtp Skipping The M1Dg Adduct To Pair With The Next Template Cytosine
Organism: Sulfolobus solfataricus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2009-06-16 Classification: TRANSFERASE Ligands: DGT, CA |
Organism: Sulfolobus solfataricus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2009-06-16
Ligands: DGT, CA
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Crystal Structure Of Vegfr2 In Complex With A 3,4,5-Trimethoxy Aniline Containing Pyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2008-10-07 Classification: TRANSFERASE Ligands: SO4, SAV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: SO4, SAV
