Search Count: 29
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Voltage-Gated Potassium Channel Kv3.1 With Novel Positive Modulator (9M)-9-{5-Chloro-6-[(3,3-Dimethyl-2,3-Dihydro-1-Benzofuran-4-Yl)Oxy]-4-Methylpyridin-3-Yl}-2-Methyl-7,9-Dihydro-8H-Purin-8-One (Compound 4)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-10-25 Classification: TRANSPORT PROTEIN Ligands: ZN, X9T, POV, K |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-10-25
Ligands: ZN, X9T, POV, K
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Voltage-Gated Potassium Channel Kv3.1 Apo
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-10-25 Classification: TRANSPORT PROTEIN Ligands: ZN, CLR, K |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-10-25
Ligands: ZN, CLR, K
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Orexin Receptor 2 (Ox2R) In Complex With G Protein And Natural Peptide-Agonist Orexin B (Oxb)
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY Release Date: 2021-02-10 Classification: MEMBRANE PROTEIN |
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY
Release Date: 2021-02-10
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Orexin Receptor 2 (Ox2R) In Complex With G Protein And Small-Molecule Agonist Compound 1
Organism: Homo sapiens, Mus musculus, Lama glama
Method: ELECTRON MICROSCOPY Release Date: 2021-02-10 Classification: MEMBRANE PROTEIN Ligands: XGD |
Organism: Homo sapiens, Mus musculus, Lama glama
Method: ELECTRON MICROSCOPY
Release Date: 2021-02-10
Ligands: XGD
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Sortilin-Progranulin Interaction With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2020-08-12 Classification: UNKNOWN FUNCTION Ligands: UMJ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: UMJ, GOL
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Sortilin-Progranulin Interaction With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2020-08-12 Classification: UNKNOWN FUNCTION Ligands: UP4, UNL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: UP4, UNL, GOL
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Sortilin-Progranulin Interaction With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2020-08-12 Classification: UNKNOWN FUNCTION Ligands: UOY, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: UOY, GOL
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Pde2 In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2018-09-19 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, EDO, FKV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: ZN, MG, EDO, FKV
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Pde2 In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2018-09-19 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, FKJ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: ZN, MG, FKJ, EDO
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Pde2 In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2018-09-19 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, FKG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: ZN, MG, FKG, EDO
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Crystal Structure Of Pde2 In Complex With Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2017-11-22 Classification: HYDROLASE Ligands: ZN, MG, CZV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-22
Ligands: ZN, MG, CZV, EDO
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Crystal Structure Of Pde2 In Complex With Complex 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2017-11-22 Classification: HYDROLASE Ligands: ZN, MG, CZY, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-22
Ligands: ZN, MG, CZY, EDO
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Pde2 In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2017-11-22 Classification: HYDROLASE Ligands: ZN, MG, D07 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-22
Ligands: ZN, MG, D07
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Identification Of Lxrbeta Selective Agonists For The Treatment Of Alzheimer'S Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-04-06 Classification: SIGNALING PROTEIN Ligands: 668, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: 668, PEG
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Identification Of Lxrbeta Selective Agonists For The Treatment Of Alzheimer'S Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2016-04-06 Classification: SIGNALING PROTEIN Ligands: 668, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: 668, SO4
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Bace1 In Complex With 4-(Cyclohexylamino)-1-(3-Fluorophenyl)-8-(3-Isopropoxybenzyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QA
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Bace1 In Complex With 8-(3-((1-Aminopropan-2-Yl)Oxy)Benzyl)-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-08-05 Classification: Hydrolase/Hydrolase inhibitor Ligands: 4QD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QD
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Bace1 In Complex With 8-Benzyl-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-7-Methyl-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QF
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The Structure Of Trka Kinase Bound To The Inhibitor N-(3-Cyclopropyl-1-Phenyl-1H-Pyrazol-5-Yl)-2-{4-[3-Methoxy-4-(4-Methyl-1H-Imidazol-1-Yl)Phenyl]-1H-1,2,3-Triazol-1-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31V, GOL, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31V, GOL, CL, ACT
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The Structure Of Trka Kinase Bound To The Inhibitor 1-Cyclopropyl-1-[3-(1,3-Thiazol-2-Yl)Benzyl]-3-[4-(Trifluoromethoxy)Phenyl]Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31W, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31W, CL, ACT