Search Count: 17
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N-Terminal Bromodomain Of Human Brd4 With (1R,1'R)-7,7'-(Ethane-1,2-Diylbis(Oxy))Bis(1,3-Dimethyl-1,3-Dihydro-2H-Benzo[D]Azepin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2023-11-08 Classification: TRANSCRIPTION Ligands: EDO, ZTT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: EDO, ZTT
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N-Terminal Bromodomain Of Human Brd4 With (1R,1'R)-7,7'-(Pentane-1,5-Diylbis(Oxy))Bis(1,3-Dimethyl-1,3-Dihydro-2H-Benzo[D]Azepin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2023-10-04 Classification: TRANSCRIPTION Ligands: ZTY, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-04
Ligands: ZTY, EDO
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N-Terminal Bromodomain Of Human Brd4 With I-Bet282
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2021-10-13 Classification: TRANSCRIPTION Ligands: EDO, UYK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: EDO, UYK
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Brd9 With 4-Chloro-2-Methyl-Methylamino-Pyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2021-04-14 Classification: TRANSCRIPTION Ligands: 82I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: 82I
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Brd9 With Biphenyl-Methylamino-Dimethylpyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2021-03-24 Classification: TRANSCRIPTION Ligands: P8W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: P8W
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Brd9 With Methylpiperazinyl-Benzyl-Amino-Dimethylpyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2021-03-24 Classification: TRANSCRIPTION Ligands: P8Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: P8Z
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N-Terminal Domain Of Brd4 With Biphenyl-Methyamino-Dimethylpyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2021-03-24 Classification: TRANSCRIPTION Ligands: P8W, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: P8W, EDO
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N-Terminal Bromodomain Of Human Brd4 With Ibet-Bd1 (Gsk778)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: GLU, LWB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: GLU, LWB, EDO
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C-Terminal Bromodomain Of Human Brd2 With Ibet-Bd1 (Gsk778)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: LWB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: LWB, EDO
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C-Terminal Bromodomain Of Human Brd2 With Ibet-Bd2 (Gsk046)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: EDO, LW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: EDO, LW5
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N-Terminal Bromodomain Of Human Brd4 With Ibet-Bd2 (Gsk046)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-01 Classification: TRANSCRIPTION Ligands: EDO, LW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: EDO, LW5
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N-Terminal Bromodomain Of Human Brd4 With I-Bet295
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2014-12-24 Classification: TRANSCRIPTION Ligands: EDO, IES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: EDO, IES
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N-Terminal Bromodomain Of Human Brd4 With Ibet-295
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-12-24 Classification: TRANSCRIPTION Ligands: EDO, 83T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: EDO, 83T
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N-Terminal Bromodomain Of Human Brd2 With I-Bet726 (Gsk1324726A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-10-08 Classification: TRANSCRIPTION Ligands: EDO, 73B, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: EDO, 73B, SO4
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C-Terminal Bromodomain Of Human Brd2 With I-Bet726 (Gsk1324726A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-10-08 Classification: TRANSCRIPTION Ligands: 73B, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 73B, SO4
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N-Terminal Bromodomain Of Human Brd2 With 1-((2R,4S)-2-Methyl-4-(Phenylamino)-6-(4-(Piperidin-1-Ylmethyl)Phenyl)-3,4-Dihydroquinolin-1(2H)-Yl)Ethanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2014-10-08 Classification: TRANSCRIPTION Ligands: 9S3, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 9S3, SO4, DMS
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With I-Bet151(Gsk1210151A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2011-11-02 Classification: SIGNALING PROTEIN Ligands: EDO, 1GH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-02
Ligands: EDO, 1GH
