Search Count: 43
![]() |
Crystal Structure Of Human Renin In Complex With A Biphenylpipderidinylcarbinol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 90D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, 90D
![]() |
Crystal Structure Of Human Renin In Complex With A Biphenylpipderidinylcarbinol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 9G7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, 9G7, SO4
![]() |
Crystal Structure Of Human Renin In Complex With A Biphenylpipderidinylcarbinol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, SO4, 9JD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, SO4, 9JD
![]() |
Crystal Structure Of Human Hexokinase 2 With Cmpd 30, A 2-Amino-6-Benzenesulfonamide Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 604 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 604
![]() |
Crystal Structure Of Human Hexokinase 2 With Cmpd 27, A 2-Amido-6-Benzenesulfonamide Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.92 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 603 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 603
![]() |
Crystal Structure Of Human Hexokinase 2 With Cmpd 1, A C-2-Substituted Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 62C, BG6, FLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 62C, BG6, FLC
![]() |
Crystal Structure Of Human Phosphorylated Ire1Alpha In Complex With A Type Iii Kinase Inhibitor (Gsk2850163A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2015-11-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4K7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: 4K7
![]() |
Crystal Structure Of Pire1Alpha In Complex With Staurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2015-11-11 Classification: Transferase/transferase inhibitor Ligands: STU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: STU
![]() |
Crystal Structure Of Human Phosphorylated Ire1Alpha In Complex With Adp-Mg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2015-11-11 Classification: TRANSFERASE Ligands: MG, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: MG, ADP
![]() |
Crystal Structure Of Human Idh1 In Complex With Gsk321A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2015-10-07 Classification: Oxidoreductase/Oxidoreductase Inhibitor Ligands: NAP, 59D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-07
Ligands: NAP, 59D
![]() |
Crystal Structure Of Cathepsin C In Complex With Dipeptide Substrates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2015-03-25 Classification: HYDROLASE Ligands: SER, TYR, NAG, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: SER, TYR, NAG, CL
![]() |
Crystal Structure Of Cathepsin C In Complex With Dipeptide Substrates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2015-03-25 Classification: HYDROLASE Ligands: GLY, LYS, SO4, NAG, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: GLY, LYS, SO4, NAG, CL, EDO
![]() |
X-Ray Structure Of Receptor Interacting Protein 1 (Rip1)Kinase Domain With A 1-Aminoisoquinoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2013-11-20 Classification: TRANSFERASE Ligands: MG, Q1A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-20
Ligands: MG, Q1A
![]() |
Crystal Structure Analysis Of Human Idh1 Mutants In Complex With Nadp+ And Ca2+/Alpha-Ketoglutarate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2013-07-31 Classification: OXIDOREDUCTASE Ligands: AKG, CA, NAP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-31
Ligands: AKG, CA, NAP
![]() |
Crystal Structure Analysis Of Human Idh1 Mutants In Complex With Nadp+ And Ca2+/Alpha-Ketoglutarate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2013-07-24 Classification: OXIDOREDUCTASE Ligands: CA, NAP, AKG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-24
Ligands: CA, NAP, AKG
![]() |
Crystal Structure Analysis Of Human Idh1 Mutants In Complex With Nadp+ And Ca2+/Alpha-Ketoglutarate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-07-17 Classification: OXIDOREDUCTASE Ligands: CA, NAP, AKG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: CA, NAP, AKG, EDO
![]() |
Crystal Structure Analysis Of Human Idh1 Mutants In Complex With Nadp+ And Ca2+/Alpha-Ketoglutarate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-07-17 Classification: OXIDOREDUCTASE Ligands: NAP, CA, EDO, AKG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: NAP, CA, EDO, AKG
![]() |
Trypsin In Complex With The Inhibitor 1-[3-(Aminomethyl)Phenyl]-N-[3-Fluoro-2'-(Methylsulfonyl)Biphenyl-4-Yl]-3-(Trifluoromethyl)-1H-Pyrazole-5-Carboxamide (Dpc423)
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-04-21 Classification: HYDROLASE Ligands: M35, CA |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2010-04-21
Ligands: M35, CA
![]() |
Factor Xa In Complex With The Inhibitor 1-[3-(Aminomethyl)Phenyl]-N-[3-Fluoro-2'-(Methylsulfonyl)Biphenyl-4-Yl]-3-(Trifluoromethyl)-1H-Pyrazole-5-Carboxamide (Dpc423)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2010-04-21 Classification: HYDROLASE Ligands: M35, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-04-21
Ligands: M35, CA
![]() |
Factor Xa In Complex With The Inhibitor 1-[2-(Aminomethyl)Phenyl]-N-(3-Fluoro-2'-Sulfamoylbiphenyl-4-Yl)-3-(Trifluoromethyl)-1H-Pyrazole-5-Carboxamide (Dpc602)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-04-21 Classification: HYDROLASE Ligands: M37, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-04-21
Ligands: M37, CA
