Search Count: 43
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Crystal Structure Of Dlk With Inhibitor Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2025-02-19 Classification: TRANSFERASE/INHIBITOR Ligands: A1AZP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1AZP
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Crystal Structure Of Dlk With Inhibitor Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2025-02-19 Classification: TRANSFERASE/INHIBITOR Ligands: A1AZ8, MG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1AZ8, MG, EDO
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Crystal Structure Of Wild Type Egfr In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2022-12-07 Classification: HYDROLASE Ligands: R28 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: R28
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Crystal Structure Of Egfr_D770_N771Insnpg/V948R In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-12-07 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: R28, EDO, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: R28, EDO, CIT
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Crystal Structure Of Human D-Amino Acid Oxidase In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-06-08 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: FAD, M7I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-08
Ligands: FAD, M7I
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Crystal Structure Of Human D-Amino Acid Oxidase In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2022-06-08 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: FAD, BEZ, M89 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-08
Ligands: FAD, BEZ, M89
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Structure Of Human Setd8 In Complex With Covalent Inhibitor Ms4138
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-05-01 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: EDO, E1J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: EDO, E1J
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Crystal Structure Of Apo Human Setd8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-03-07 Classification: TRANSFERASE Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: EDO
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Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With Hinge Binding Pyrazolobenzothiazine Compound.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2013-03-06 Classification: transferase/transferase inhibitor Ligands: 1BQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: 1BQ
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Crystal Structure Of Human Dipeptidyl Peptidase Iv In Complex With A Pyridopyrimidinedione Analogue
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-02-27 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0WG, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-27
Ligands: 0WG, NAG
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Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With An Allosteric Binding Pyrazolobenzothiazine Compound.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2013-02-06 Classification: transferase/transferase inhibitor Ligands: IPA, 1BR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-06
Ligands: IPA, 1BR
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Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With Novel Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2012-08-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0O7, IPA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-22
Ligands: 0O7, IPA
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Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With Novel Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2012-07-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0PF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-25
Ligands: 0PF
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With Tak-322
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, T22 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: NAG, T22
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With A Pyrimidinedione Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: RUF, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: RUF, NAG
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With A Pyrimidinedione Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: XIH, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: XIH, NAG
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With A Pyrimidinone Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2010-02-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: RUM, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: RUM, NAG
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Crystal Structure Of Human Dpp4 In Complex With A Benzimidazole Derivative
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2008-10-21 Classification: HYDROLASE Ligands: NAG, B2Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-21
Ligands: NAG, B2Y
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Crystal Structure Of Human Dpp4 In Complex With A Benzimidazole Derivative
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2008-10-21 Classification: HYDROLASE Ligands: NAG, 7AC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-21
Ligands: NAG, 7AC
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Crystal Structure Of Human Dpp-4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2008-03-04 Classification: HYDROLASE Ligands: NAG, SY1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-04
Ligands: NAG, SY1
