Search Count: 84
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Crystal Structure Of Cbl-B Tkb Bound To Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2024-07-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, A1AEG, GOL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: MG, A1AEG, GOL, PEG
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Crystal Structure Of Cbl-B Tkb Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2024-07-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, CA, A1AD4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: MG, CA, A1AD4
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Pcsk9-Fab 7G7 Complex Bound To Cis-1-Amino-4-Phenylcyclohexaneacyl-Wnlk(Hr)Igllr - Nh2
Organism: Homo sapiens, Mus musculus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.94 Å Release Date: 2020-02-05 Classification: HYDROLASE/HYDROLASE INHIBITOR/IMMUNE SYSTEM Ligands: CA |
Organism: Homo sapiens, Mus musculus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-02-05
Ligands: CA
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Design Of Organo-Peptides As Bipartite Pcsk9 Antagonists
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2020-02-05 Classification: HYDROLASE/HYDROLASE INHIBITOR/IMMUNE SYSTEM Ligands: CA |
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2020-02-05
Ligands: CA
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Pcsk9 Complex With Fab33
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2017-08-16 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
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Short Pcsk9 Delta-P' Complex With Fusion2 Peptide
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-08-16 Classification: HYDROLASE Ligands: CA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: CA
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Short Pcsk9 Delta-P' Complex With Peptide Pep1
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2017-08-16 Classification: HYDROLASE Ligands: CA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: CA
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Short Pcsk9 Delta-P' Complex With Shrunken Peptide Bearing Homo-Arginine
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-08-16 Classification: HYDROLASE Ligands: CA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: CA
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Short Pcsk9 Delta-P' Complex With Peptide Pep3
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2017-08-16 Classification: HYDROLASE Ligands: CA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: CA
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Pcsk9 Complex With Ldlr Antagonist Peptide And Fab7G7
Organism: Homo sapiens, Mus musculus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-08-16 Classification: HYDROLASE |
Organism: Homo sapiens, Mus musculus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
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Crystal Structure Of The Apo-Form Of Usp7 Catalytic Domain [V302K] Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-08-09 Classification: HYDROLASE Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: GOL
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Crystal Structure Of Usp7 Catalytic Domain [V302K] Mutant In Complex With Ubiquitin (Malonate Bound)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2017-08-09 Classification: HYDROLASE Ligands: MLA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: MLA, GOL
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Crystal Structure Of Usp7 Catalytic Domain [V302K] Mutant In Complex With Ubiquitin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2017-08-09 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
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Crystal Structure Of Usp7 Catalytic Domain [H294E] Mutant In Complex With Ubiquitin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2017-08-09 Classification: HYDROLASE Ligands: EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: EPE
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Crystal Structure Of Usp7 Catalytic Domain [L299A] Mutant In Complex With Ubiquitin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2017-08-09 Classification: HYDROLASE Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: GOL
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Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Sorafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BAX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: BAX
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Egfr Kinase Domain Mutant "Tmlr" With A Pyrazolopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 63M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: 63M
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Egfr Kinase Domain Mutant "Tmlr" With A Imidazopyridinyl-Aminopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 63N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: SO4, 63N
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Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Az628
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B1E, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: B1E, PEG
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Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Dabrafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P06 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: P06
