Search Count: 22
![]() |
Crystal Structure Of Mdm2 With Brigimadlin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2024-10-02 Classification: LIGASE Ligands: G7I |
![]() |
Crystal Structure Of Human Syk In Complex With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-04-24 Classification: TRANSFERASE Ligands: A1H2W, GOL |
![]() |
Crystal Structure Of Syk Kinase In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2024-04-24 Classification: TRANSFERASE Ligands: A1H2Y, GOL |
![]() |
Crystal Structure Of The Legionella Pneumophila Chia C-Terminal Domain
Organism: Legionella pneumophila 130b
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2020-04-22 Classification: SUGAR BINDING PROTEIN Ligands: MPD, MRD |
![]() |
The Catalytic Fragment Of Poly(Adp-Ribose) Polymerase Complexed With Isoindolinone Inhibitor
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: H7W |
![]() |
The Catalytic Fragment Of Poly(Adp-Ribose) Polymerase Complexed With An Isoindolinone Inhibitor
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: H7Z |
![]() |
Crystal Structure Of Aurora B In Complex With Bi 847325
Organism: Xenopus laevis
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2016-08-17 Classification: TRANSFERASE Ligands: 5U5 |
![]() |
Mek1 In Complex With Bi 847325
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-08-17 Classification: TRANSFERASE Ligands: 5U5, CA |
![]() |
Crystal Structure Of Aurorab/Incenp In Complex With Bi 811283
Organism: Xenopus laevis
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-08-17 Classification: TRANSFERASE Ligands: 6Q4 |
![]() |
Crystal Structure Of The Alk Kinase Domain In Complex With Entrectinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2016-04-06 Classification: TRANSFERASE Ligands: YMX |
![]() |
Crystal Structure Of The Alk Kinase Domain In Complex With Cmpd 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-04-06 Classification: TRANSFERASE Ligands: U4W, GOL |
![]() |
Structure Of Parp2 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: FSU |
![]() |
Structure Of Human Parp2 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: D7N |
![]() |
Structure Of Human Parp1 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: SO4, GOL, FSU |
![]() |
Structure Of Human Parp1 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: D7N, SO4 |
![]() |
Structure Of Human Anaplastic Lymphoma Kinase In Complex With Nvp- Tae684
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-07-28 Classification: TRANSFERASE Ligands: GUI |
![]() |
Structure Of Human Anaplastic Lymphoma Kinase In Complex With Pha- E429
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2010-07-28 Classification: TRANSFERASE Ligands: 571 |
![]() |
Optimisation Of 6,6-Dimethyl Pyrrolo 3,4-C Pyrazoles: Identification Of Pha-793887, A Potent Cdk Inhibitor Suitable For Intravenous Dosing
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2010-02-23 Classification: CELL CYCLE Ligands: SO4, 889 |
![]() |
Crystal Structure Of Gsk-3 Beta In Complex With Nms-869553A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-03-03 Classification: TRANSFERASE Ligands: 553 |
![]() |
Structure Of Cdk2-Cyclin A With Pha-630529
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2005-12-08 Classification: TRANSFERASE Ligands: 529, SO4 |




















