Search Count: 47
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Brain Penetrant Liver X Receptor (Lxr) Modulators Based On A 2,4,5,6-Tetrahydropyrrolo[3,4-C]Pyrazole Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-21 Classification: DNA BINDING PROTEIN Ligands: 6Y4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6Y4
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Brain Penetrant Liver X Receptor (Lxr) Modulators Based On A 2,4,5,6-Tetrahydropyrrolo[3,4-C]Pyrazole Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-09-21 Classification: DNA BINDING PROTEIN Ligands: 6Y8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6Y8
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Discovery Of Novel, Orally Efficacious Liver X Receptor (Lxr) Beta Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2016-06-29 Classification: DNA BINDING PROTEIN Ligands: 67S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: 67S
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Identification Of Spirooxindole And Dibenzoxazepine Motifs As Potent Mineralocorticoid Receptor Antagonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-03-09 Classification: SIGNALING PROTEIN Ligands: 60R, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-09
Ligands: 60R, CL
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Crystal Structure Of S.A. Gyrase In Complex With Compound 7
Organism: Staphylococcus aureus, Staphylococcus aureus subsp. aureus ed98
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-06-17 Classification: Isomerase/DNA/RNA Ligands: MN, SO4, WCP |
Organism: Staphylococcus aureus, Staphylococcus aureus subsp. aureus ed98
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: MN, SO4, WCP
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Crystal Structure Of Staph Gyraseb 24Kda In Complex With Kibdelomycin
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:2.94 Å Release Date: 2014-07-30 Classification: ISOMERASE Ligands: XAM |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: XAM
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Crystal Structure Of Staph Gyraseb 24Kda In Complex With Novobiocin
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2014-07-30 Classification: ISOMERASE Ligands: NOV |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: NOV
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Crystal Structure Of Staph Pare43Kda In Complex With Kbd
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2014-07-16 Classification: ISOMERASE Ligands: XAM |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-07-16
Ligands: XAM
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Crystal Structure Of Staph Pare 24Kda In Complex With Novobiocin
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-07-16 Classification: ISOMERASE Ligands: NOV |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-07-16
Ligands: NOV
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Crystal Structure Of S.A. Gyrase-Am8191 Complex
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2014-06-18 Classification: ISOMERASE/ISOMERASE Inhibitor/DNA Ligands: 31N, SO4, MN |
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31N, SO4, MN
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Structure Of Lpxc Bound To The Reaction Product Udp-(3-O-(R-3-Hydroxymyristoyl))-Glucosamine
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2013-10-16 Classification: HYDROLASE Ligands: ZN, 24G, PO4 |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2013-10-16
Ligands: ZN, 24G, PO4
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Crystal Structure Of Ribosome Inactivating Protein From Momordica Balsamina Complexed With The Product Of Rna Substrate Adenosine Triphosphate At 2.0 A Resolution
Organism: Momordica balsamina
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2012-01-18 Classification: HYDROLASE Ligands: NAG, GOL, ADE |
Organism: Momordica balsamina
Method: X-RAY DIFFRACTION
Release Date: 2012-01-18
Ligands: NAG, GOL, ADE
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Crystal Structure Of The Complex Formed Between Type 1 Ribosome Inactivating Protein And Adenine At 1.7A Resolution
Organism: Momordica balsamina
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2011-12-07 Classification: HYDROLASE Ligands: NAG, ADE, GOL |
Organism: Momordica balsamina
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: NAG, ADE, GOL
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Clinically Useful Alkyl Amine Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2011-11-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, CL, RX5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-30
Ligands: NAG, CL, RX5
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Clinically Useful Alkyl Amine Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2011-11-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CL, RX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-30
Ligands: CL, RX6
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Alkyl Amine Renin Inhibitors: Filling S1 From S3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-08-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: RX0, GOL, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-03
Ligands: RX0, GOL, NAG
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Crystal Structure Of The Complex Of Type I Ribosome Inactivating Protein From Momordica Balsamina With 5-(Hydroxymethyl)Oxalane-2,3,4-Triol At 1.6 A Resolution
Organism: Momordica balsamina
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2011-08-03 Classification: HYDROLASE Ligands: NAG, RIP, GOL |
Organism: Momordica balsamina
Method: X-RAY DIFFRACTION
Release Date: 2011-08-03
Ligands: NAG, RIP, GOL
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Crystal Structure Of Native Type 1 Ribosome Inactivating Protein From Momordica Balsamina At 1.67 A Resolution
Organism: Momordica balsamina
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2011-07-06 Classification: HYDROLASE Ligands: NAG, GOL |
Organism: Momordica balsamina
Method: X-RAY DIFFRACTION
Release Date: 2011-07-06
Ligands: NAG, GOL
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Crystal Structure Of The Complex Of Type I Rip With The Hydrolyzed Product Of Datp, Adenine At 1.9 A Resolution
Organism: Momordica balsamina
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-05-11 Classification: HYDROLASE Ligands: NAG, GOL, ADE |
Organism: Momordica balsamina
Method: X-RAY DIFFRACTION
Release Date: 2011-05-11
Ligands: NAG, GOL, ADE
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Crystal Structure Of E. Coli Fabf(C163A) In Complex With Platensimycin A1
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-07-28 Classification: TRANSFERASE Ligands: 840 |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2010-07-28
Ligands: 840
