Search Count: 20
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Crystal Structure Of Human Ripk1 With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2025-05-28 Classification: TRANSFERASE/INHIBITOR Ligands: A1BU4, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1BU4, IOD
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Crystal Structure Of Human Ripk1 With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2025-05-28 Classification: TRANSFERASE/INHIBITOR Ligands: A1BU6, IOD, GLY, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1BU6, IOD, GLY, CL
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Crystal Structure Of Ripk1 With Compound 36
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2025-05-28 Classification: TRANSFERASE/INHIBITOR Ligands: A1BU5, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1BU5, IOD
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Co-Crystal Structure Of Human Prmt9 In Complex With Mrk-990 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2024-12-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1AHM, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1AHM, UNX
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Co-Crystal Structure Of Human Carm1 In Complex With Mt556 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-01-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 44T, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: 44T, UNX
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Co-Crystal Structure Of Human Prmt9 In Complex With Mt221 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2021-12-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EJB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-22
Ligands: EJB
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Human Arginase1 Complexed With Inhibitor Compound 3A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2021-09-29 Classification: HYDROLASE/INHIBITOR Ligands: MN, XFP, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: MN, XFP, EDO
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Human Arginase1 Complexed With Inhibitor Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2021-09-29 Classification: HYDROLASE/INHIBITOR Ligands: MN, XFG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: MN, XFG
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Human Arginase1 Complexed With Inhibitor Compound 24A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2021-09-29 Classification: HYDROLASE/INHIBITOR Ligands: MN, 0IZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: MN, 0IZ
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Co-Crystal Structure Of Human Prmt9 In Complex With Mt556 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-08-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 44T, EDO, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: 44T, EDO, UNX
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Prmt5:Mep50 Complexed With 5,5-Bicyclic Inhibitor Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: WFM, EDO, CL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: WFM, EDO, CL, PEG
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Prmt5:Mep50 Complexed With 5,5-Bicyclic Inhibitor Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EDO, WFS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: EDO, WFS
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Prmt5:Mep50 Complexed With 5,5-Bicyclic Inhibitor Compound 72
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EDO, WFV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: EDO, WFV
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Hpk1 In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2021-03-17 Classification: TRANSFERASE Ligands: XHV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-17
Ligands: XHV
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Hpk1 In Complex With Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-03-17 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: XHS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-17
Ligands: XHS, EDO
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Hpk1 In Complex With Compound 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-03-17 Classification: TRANSFERASE Ligands: XHM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-17
Ligands: XHM
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Crystal Structure Of The Human Leukotriene B4 Receptor 1 In Complex With Selective Antagonist Mk-D-046
Organism: Homo sapiens, Desulfovibrio vulgaris (strain hildenborough / atcc 29579 / dsm 644 / ncimb 8303)
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2021-02-17 Classification: MEMBRANE PROTEIN Ligands: VRJ, NA, FMN, OLA, OLC, 1PE, 2PE, P6G |
Organism: Homo sapiens, Desulfovibrio vulgaris (strain hildenborough / atcc 29579 / dsm 644 / ncimb 8303)
Method: X-RAY DIFFRACTION
Release Date: 2021-02-17
Ligands: VRJ, NA, FMN, OLA, OLC, 1PE, 2PE, P6G
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Prmt5:Mep50 Complexed With Allosteric Inhibitor Compound 1A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2020-08-19 Classification: TRANSFERASE/Transcription Ligands: QL1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: QL1
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Prmt5:Mep50 Complexed With Allosteric Inhibitor Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2020-08-19 Classification: TRANSFERASE/TRANSCRIPTION Ligands: QKY, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: QKY, EDO, GOL
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Discovery Of 1-1H-Pyrazolo 4,3-C Pyridine-6-Yl Urea Inhibitors Of Extracellular Signal Regulated Kinase Erk For The Treatment Of Cancers
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2016-07-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6S9, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 6S9, SO4
