Search Count: 18
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Crystal Structure Of Wild-Type Egfr In Complex With The Reversible Inhibitor Sevabertinib (Bay 2927088)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2025-10-15 Classification: TRANSFERASE Ligands: SIN, CL, DMS, EDO, A1JBI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-15
Ligands: SIN, CL, DMS, EDO, A1JBI
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q2X, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q2X, GOL
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Crystal Structure Of Pparg And Ncor2 With Sr10221, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: A8R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: A8R
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q33 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q33
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Crystal Structure Of Mutant Pparg (C313A) And Ncor2 With An Inverse Agonist (Compound 7E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q33 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q33
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7D)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q1R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q1R
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Crystal Structure Of Mutant Pparg (C313A) And Ncor2 With An Inverse Agonist (Compound Si-1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q4O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q4O
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound Si-2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q5X, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q5X, SO4
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 15B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q8F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q8F
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Crystal Structure Of Pparg And Ncor2 With Bay-5516, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q5O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q5O
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Crystal Structure Of Pparg And Ncor2 With Bay-9683, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q4C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: Q4C
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X-Ray Structure Of Smyd3 In Complex With Benzodiazepine-Type Inhibitor Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZT, SAM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZT, SAM, ZN
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X-Ray Structure Of Smyd3 In Complex With Benzodiazepine-Type Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZQ, ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZQ, ZN, SAM
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X-Ray Structure Of Smyd3 In Complex With The Benzodiazepine-Based Probe Bay-6035
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZK, SAM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZK, SAM, ZN
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Lytr-Csp2A-Psr Enzyme From Actinomyces Oris
Organism: Actinomyces oris
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2018-04-11 Classification: TRANSCRIPTION Ligands: CO, PO4, PE4 |
Organism: Actinomyces oris
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: CO, PO4, PE4
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Crystal Structure Of The Second Bromodomain Of Human Taf1 In Complex With Bay-299 Chemical Probe
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2017-05-03 Classification: TRANSCRIPTION Ligands: EDO, 7M8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-03
Ligands: EDO, 7M8
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Brpf2 In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2017-05-03 Classification: TRANSCRIPTION Ligands: 8LW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-03
Ligands: 8LW
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Srta Sortase From Actinomyces Oris
Organism: Actinomyces oris
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2017-03-01 Classification: HYDROLASE Ligands: CL |
Organism: Actinomyces oris
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: CL
