Search Count: 79
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Crystal Structure Of Pi3K-Alpha In Complex With Taselisib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: 799 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: 799
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3W
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3R
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3N
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Lactate Dehydrogenase In Complex With Inhibitor 6-(3-Aminophenyl)-3-((2-Chlorophenyl)Thio)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, EPE, SO4, D4S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, EPE, SO4, D4S
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Lactate Dehydrogenase In Complex With Inhibitor (S)-5-((2-Chlorophenyl)Thio)-6'-((4-Fluorophenyl)Amino)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: EPE, NAD, LAC, SO4, D47 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: EPE, NAD, LAC, SO4, D47
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Lactate Dehydrogenase In Complex With Inhibitor (R)-3-((2-Chlorophenyl)Thio)-6-(3-((4-Fluorophenyl)Amino)Phenyl)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE Ligands: NAD, EPE, SO4, D3S, LAC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, EPE, SO4, D3S, LAC
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Lactate Dehydrogenase In Complex With Inhibitor (R)-5-((2-Chlorophenyl)Thio)-6'-(4-Fluorophenoxy)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, SO4, D3J, LAC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, SO4, D3J, LAC
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Lactate Dehydrogenase In Complex With Inhibitor (S)-5-((2-Chlorophenyl)Thio)-6'-(4-Fluorophenoxy)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, SO4, LAC, D4J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, SO4, LAC, D4J
 |
Lactate Dehydrogenase In Complex With Inhibitor 3-((2-Chlorophenyl)Thio)-6-(6-((4-Fluorophenyl)Amino)Pyridin-2-Yl)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, SO4, D4A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, SO4, D4A
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Lactate Dehydrogenase In Complex With Inhibitor (R)-3-((2-Chlorophenyl)Thio)-6-(3-((4-Fluorophenyl)Amino)Phenyl)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-10-17 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, EPE, SO4, D0Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: NAD, EPE, SO4, D0Y
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Lactate Dehydrogenase In Complex With Inhibitor (R)-5-((2-Chlorophenyl)Thio)-6'-((4-Fluorophenyl)Amino)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-10-17 Classification: OXIDOREDUCTASE/Inhibitor Ligands: EPE, NAD, SO4, D0V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: EPE, NAD, SO4, D0V
 |
Lactate Dehydrogenase In Complex With Hydroxylactam Inhibitor Compound 9: (6R)-3-[(2-Chlorophenyl)Sulfanyl]-4-Hydroxy-6-(3-Hydroxyphenyl)-6-(Thiophen-3-Yl)-5,6-Dihydropyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2016-09-14 Classification: OXIREDUCTASE/OXIREDUCTASE INHIBITOR Ligands: EPE, TXD, 6EY, SO4, NAI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: EPE, TXD, 6EY, SO4, NAI
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Lactate Dehydrogenase In Complex With Hydroxylactam Inhibitor Compound 31: (2~{S})-5-(2-Chlorophenyl)Sulfanyl-2-(4-Morpholin-4-Ylphenyl)-4-Oxidanyl-2-Thiophen-3-Yl-1,3-Dihydropyridin-6-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-09-14 Classification: OXIREDUCTASE/OXIREDUCTASE INHIBITOR Ligands: NAD, SO4, GN2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: NAD, SO4, GN2
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Egfr Kinase Domain Mutant "Tmlr" With Azabenzimidazole Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60B
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Egfr Kinase Domain Mutant "Tmlr" With 3-Carboxamide Azaindole Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60D
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Egfr Kinase Domain Mutant "Tmlr" With 3-Azetidinyl Azaindazole Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60E
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Lactate Dehydrogenase A In Complex With A Trisubstituted Piperidine-2,4-Dione Inhibitor Gne-140
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-18 Classification: Oxidoreductase/Oxidoreductase Inhibitor Ligands: NAD, SO4, GN0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: NAD, SO4, GN0
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P110Alpha/P85Alpha With Compound 5
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-01-27 Classification: Transferase/Transferase Inhibitor Ligands: 5H2 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H2
 |
P110Alpha With Gdc-0326
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2016-01-27 Classification: Transferase/Inhibitor Ligands: 5H5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H5, EDO