Search Count: 26
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Il17A Homodimer Complexed To Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCE
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Il17A Complexed To Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCW, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCW, CL
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Crystal Structure Of Hpk1 (Map4K1) Complex With Inhibitor A-745
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2022-03-02 Classification: SIGNALING PROTEIN, Transferase Ligands: 9ID, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-02
Ligands: 9ID, SO4
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Hcv Ns5B 1B N316 Bound To Compound 18
Organism: Hepatitis c virus subtype 1b
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-09-04 Classification: VIRAL PROTEIN Ligands: K4J |
Organism: Hepatitis c virus subtype 1b
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: K4J
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Hcv Ns5B 1A Y316 Bound To Compound 49
Organism: Hepacivirus c
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2019-09-04 Classification: VIRAL PROTEIN Ligands: SO4, K4P |
Organism: Hepacivirus c
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: SO4, K4P
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Hcv Ns5B 1B N316 Bound To Compound 18
Organism: Hepatitis c virus genotype 1b (isolate bk)
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-09-04 Classification: VIRAL PROTEIN Ligands: K4S |
Organism: Hepatitis c virus genotype 1b (isolate bk)
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: K4S
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Hcv Ns5B 1B N316 Bound To Compound 31
Organism: Hepatitis c virus subtype 1b
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2019-09-04 Classification: VIRAL PROTEIN Ligands: K4M |
Organism: Hepatitis c virus subtype 1b
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: K4M
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Crystal Structure Of Il-36Gamma Complexed To A-552
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-06-26 Classification: CYTOKINE Ligands: O6D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: O6D
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Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: CA, ICT, DWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: CA, ICT, DWP
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Novel Binding Modes Of Inhibition Of Wild-Type Idh1: Allosteric Inhibition With Cmpd2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: LMR, MG, K32 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: LMR, MG, K32
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Novel Modes Of Inhibition Of Wild-Type Idh1: Non-Equivalent Allosteric Inhibition With Cmpd3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, DWM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: NAP, DWM
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Novel Modes Of Inhibition Of Wild-Type Idh1:Direct Covalent Modification Of His315 With Cmpd11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: MG, ICT, DWJ, NAP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: MG, ICT, DWJ, NAP
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Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: ICT, DWG, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: ICT, DWG, CA
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Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: CA, ICT, DWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: CA, ICT, DWS
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The Structure Of Human Pde12 Residues 161-609
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2015-06-17 Classification: HYDROLASE Ligands: MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: MG, GOL
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The Structure Of Human Pde12 Residues 161-609 In Complex With Gsk3036342A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-06-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: SO4, EDO, TRS, 4LC, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: SO4, EDO, TRS, 4LC, MG
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Hcv Ns5B Gt1A C316Y With Gsk5852
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2013-05-29 Classification: REPLICATION/REPLICATION INHIBITOR Ligands: SO4, 1PV |
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: SO4, 1PV
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Hcv Ns5B Gt1B N316Y With Gsk5852
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2013-05-15 Classification: REPLICATION/REPLICATION INHIBITOR Ligands: 1PV |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2013-05-15
Ligands: 1PV
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Hcv Ns5B Gt1A With Gsk5852
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-05-15 Classification: REPLICATION/REPLICATION INHIBITOR Ligands: 1PV, SO4 |
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION
Release Date: 2013-05-15
Ligands: 1PV, SO4
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Hcv Ns5B Gt1B N316 With Gsk5852A
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-05-08 Classification: REPLICATION/REPLICATION INHIBITOR Ligands: 1PV |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2013-05-08
Ligands: 1PV
