Search Count: 36
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Il17A Homodimer Complexed To Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCE
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Il17A Complexed To Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCW, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCW, CL
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Crystal Structure Of Hpk1 (Map4K1) Complex With Inhibitor A-745
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2022-03-02 Classification: SIGNALING PROTEIN, Transferase Ligands: 9ID, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-02
Ligands: 9ID, SO4
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Hcv Ns5B 1B N316 Bound To Compound 18
Organism: Hepatitis c virus subtype 1b
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-09-04 Classification: VIRAL PROTEIN Ligands: K4J |
Organism: Hepatitis c virus subtype 1b
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: K4J
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Hcv Ns5B 1A Y316 Bound To Compound 49
Organism: Hepacivirus c
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2019-09-04 Classification: VIRAL PROTEIN Ligands: SO4, K4P |
Organism: Hepacivirus c
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: SO4, K4P
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Hcv Ns5B 1B N316 Bound To Compound 18
Organism: Hepatitis c virus genotype 1b (isolate bk)
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-09-04 Classification: VIRAL PROTEIN Ligands: K4S |
Organism: Hepatitis c virus genotype 1b (isolate bk)
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: K4S
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Hcv Ns5B 1B N316 Bound To Compound 31
Organism: Hepatitis c virus subtype 1b
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2019-09-04 Classification: VIRAL PROTEIN Ligands: K4M |
Organism: Hepatitis c virus subtype 1b
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: K4M
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Crystal Structure Of Il-36Gamma Complexed To A-552
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-06-26 Classification: CYTOKINE Ligands: O6D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: O6D
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Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: CA, ICT, DWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: CA, ICT, DWP
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Novel Binding Modes Of Inhibition Of Wild-Type Idh1: Allosteric Inhibition With Cmpd2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: LMR, MG, K32 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: LMR, MG, K32
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Novel Modes Of Inhibition Of Wild-Type Idh1: Non-Equivalent Allosteric Inhibition With Cmpd3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, DWM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: NAP, DWM
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Novel Modes Of Inhibition Of Wild-Type Idh1:Direct Covalent Modification Of His315 With Cmpd11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2018-07-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: MG, ICT, DWJ, NAP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: MG, ICT, DWJ, NAP
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Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: ICT, DWG, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: ICT, DWG, CA
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Novel Modes Of Inhibition Of Wild-Type Idh1: Direct Covalent Modification Of His315 With Cmpd15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2018-07-25 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: CA, ICT, DWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: CA, ICT, DWS
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Crystal Structure Of The Atp Binding Domain Of S. Aureus Gyrb Complexed With A Fragment
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2016-02-03 Classification: ISOMERASE/ISOMERASE INHIBITOR Ligands: EVO, SO4, MPD |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: EVO, SO4, MPD
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Crystal Structure Of The Atp Binding Domain Of S. Aureus Gyrb Complexed With A Fragment
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2016-02-03 Classification: ISOMERASE Ligands: MPD, CL, 54X, MG |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: MPD, CL, 54X, MG
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Crystal Structure Of The Atp Binding Domain Of S. Aureus Gyrb Complexed With A Fragment
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2016-02-03 Classification: ISOMERASE/ISOMERASE INHIBITOR Ligands: 55D, MG, CL, MPD |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 55D, MG, CL, MPD
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Crystal Structure Of The Atp Binding Domain Of S. Aureus Gyrb Complexed With A Fragment
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-02-03 Classification: ISOMERASE/ISOMERASE INHIBITOR Ligands: MPD, 55G, MG |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: MPD, 55G, MG
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Crystal Structure Of The Atp Binding Domain Of S. Aureus Gyrb Complexed With A Fragment
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-02-03 Classification: ISOMERASE/ISOMERASE INHIBITOR Ligands: MPD, CL, MG, 55H |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: MPD, CL, MG, 55H
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Crystal Structure Of The Atp Binding Domain Of S. Aureus Gyrb Complexed With A Ligand
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2015-11-25 Classification: ISOMERASE/ISOMERASE INHIBITOR Ligands: 57U, MPD, GOL |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2015-11-25
Ligands: 57U, MPD, GOL
