Search Count: 23
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G9A In Complex With Rk-133232 (Compound 16G)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2025-05-21 Classification: TRANSFERASE Ligands: ZN, SFG, A1L57 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-21
Ligands: ZN, SFG, A1L57
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G9A In Complex With The S-Isomer Of Rk-131902 (Racemic Compound Rac-10A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2025-05-21 Classification: TRANSFERASE Ligands: ZN, SFG, A1L58 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-21
Ligands: ZN, SFG, A1L58
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Structure Of G9A In Complex With Compound 7I
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2025-01-22 Classification: TRANSFERASE Ligands: ZN, SFG, A1L07 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: ZN, SFG, A1L07
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Structure Of G9A In Complex With Compound 9A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2025-01-22 Classification: TRANSFERASE Ligands: ZN, SFG, A1L08 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: ZN, SFG, A1L08
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Structure Of G9A In Complex With Compound 9B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2025-01-22 Classification: TRANSFERASE Ligands: ZN, SFG, A1L09 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: ZN, SFG, A1L09
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Structure Of G9A In Complex With Compound 10A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2023-03-29 Classification: TRANSFERASE Ligands: ZN, SFG, I5X, TRS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-29
Ligands: ZN, SFG, I5X, TRS, EDO
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Structure Of G9A In Complex With Compound 10D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-03-29 Classification: TRANSFERASE Ligands: ZN, SFG, I6L, EDO, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-29
Ligands: ZN, SFG, I6L, EDO, TRS
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Structure Of G9A In Complex With Compound 11A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2023-03-29 Classification: TRANSFERASE Ligands: ZN, SFG, I6S, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-29
Ligands: ZN, SFG, I6S, EDO, CL
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Structure Of G9A In Complex With Compound 26A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2023-03-29 Classification: TRANSFERASE Ligands: ZN, CL, SFG, I6Z, EDO, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-29
Ligands: ZN, CL, SFG, I6Z, EDO, TRS
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Structure Of G9A In Complex With Rk-701
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2022-12-21 Classification: TRANSFERASE Ligands: ZN, SFG, J26, EDO, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-21
Ligands: ZN, SFG, J26, EDO, TRS
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Tankyrase-2 In Complex With Rk-582
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-04-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DU9, ZN, PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: DU9, ZN, PO4, GOL
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Tankyrase-2 In Complex With Compound 1A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2019-04-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 9GX, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: ZN, 9GX, SO4, GOL
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Tankyrase-2 In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2019-04-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 9H3, PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: ZN, 9H3, PO4, GOL
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Tankyrase-2 In Complex With Compound 52
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2019-04-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 9H6, PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: ZN, 9H6, PO4, GOL
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Tankyrase-2 In Complex With Compound 40C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2019-04-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 9H9, PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: ZN, 9H9, PO4, GOL
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Tankyrase-2 In Complex With Compound 15D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2019-04-03 Classification: TRANSFERASE Ligands: ZN, 9SU, PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: ZN, 9SU, PO4, GOL
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Crystal Structure Of Hck Complexed With A Pyrrolo-Pyrimidine Inhibitor (S)-2-(((1R,4S)-4-(4-Amino-5-(4-Phenoxyphenyl)-7H-Pyrrolo[2,3-D]Pyrimidin-7-Yl)Cyclohexyl)Amino)-4-Methylpentanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2017-10-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OOQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-11
Ligands: OOQ
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Crystal Structure Of Hck Complexed With A Pyrrolo-Pyrimidine Inhibitor (S)-Ethyl2-(((1R,4S)-4-(4-Amino-5-(4-Phenoxyphenyl)-7H-Pyrrolo[2,3-D]Pyrimidin-7-Yl)Cyclohexyl)Amino)-4-Methylpentanoate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-10-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OOO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: OOO
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Crystal Structure Of Hck Complexed With A Pyrrolo-Pyrimidine Inhibitor (S)-2-(((1R,4S)-4-(4-Amino-5-(4-Phenoxyphenyl)-7H-Pyrrolo[2,3-D]Pyrimidin-7-Yl)Cyclohexyl)Amino)-4-Methylpentanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2017-10-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OOS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: OOS
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Crystal Structure Of Hck Complexed With A Pyrrolo-Pyrimidine Inhibitor (S)-2-(((1R,4S)-4-(4-Amino-5-(4-Phenoxyphenyl)-7H-Pyrrolo[2,3-D]Pyrimidin-7-Yl)Cyclohexyl)Amino)-N,4-Dimethylpentanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-10-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OOU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: OOU
