Search Count: 10
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Crystal Structure Of An Mkp5 Mutant, Y435F, In Complex With An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2025-07-30 Classification: HYDROLASE/INHIBITOR Ligands: CJA, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-30
Ligands: CJA, SO4
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Crystal Structure Of An Mkp5 Mutant, Y435W, In Complex With An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2025-05-28 Classification: HYDROLASE/INHIBITOR Ligands: CJA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CJA
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Crystal Structure Of The Allosteric Mkp5 Mutant Y435W
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-05-14 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
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Structure Of Map Kinase Phosphatase 5 In Complex With 3,3-Dimethyl-1-((9-Propyl-5,6-Dihydrothieno[3,4-H]Quinazolin-2-Yl)Thio)Butan-2-One, An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-10-05 Classification: HYDROLASE/INHIBITOR Ligands: L8K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: L8K
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Structure Of Map Kinase Phosphatase 5 In Complex With 3,3-Dimethyl-1-((9-Propyl-5,6-Dihydrothieno[2,3-H]Quinazolin-2-Yl)Thio)Butan-2-One, An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.14 Å Release Date: 2022-10-05 Classification: HYDROLASE/INHIBITOR Ligands: L8R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: L8R
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Structure Of Map Kinase Phosphatase 5 In Complex With 3,3-Dimethyl-1-((5,6-Dihydrobenzo[H]Quinazolin-2-Yl)Thio)Butan-2-One, An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2022-10-05 Classification: HYDROLASE/INHIBITOR Ligands: NUN, DTT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: NUN, DTT
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Structure Of Map Kinase Phosphatase 5 In Complex With 3,3-Dimethyl-1-((5,6-Dihydropyrido[2,3-H]Quinazolin-2-Yl)Thio)Butan-2-One, An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-10-05 Classification: HYDROLASE/INHIBITOR Ligands: NUU, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: NUU, ACT
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Structure Of Map Kinase Phosphatase 5 In Complex With 3,3-Dimethyl-1-((9-Chloro-5,6-Dihydrobenzo[H]Quinazolin-2-Yl)Thio)Butan-2-One, An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2022-10-05 Classification: HYDROLASE/INHIBITOR Ligands: NV3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: NV3
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Structure Of Map Kinase Phosphatase 5 In Complex With 3,3-Dimethyl-1-((9-Propyl-5,6-Dihydrothieno[3,4-H]Quinazolin-2-Yl)Thio)Butan-2-One, An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2022-10-05 Classification: HYDROLASE/INHIBITOR Ligands: NVF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: NVF
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Structure Of Map Kinase Phosphatase 5 In Complex With 3,3-Dimethyl-1-((9-(Methylthio)-5,6-Dihydrothieno[3,4-H]Quinazolin-2-Yl)Thio)Butan-2-One, An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2020-08-19 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CJA, DTT, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: CJA, DTT, ACT
