Search Count: 9
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Discovery Of Mk-8353: An Orally Bioavailable Dual Mechanism Erk Inhibitor For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, G67 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SO4, G67
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Discovery Of 3(S)-Thiomethyl Pyrrolidine Erk Inhibitors For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-05-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SO4, F8V |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: SO4, F8V
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Gpr40 In Complex With Partial Agonist Mk-8666
Organism: Homo sapiens, Enterobacteria phage t4
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-06-07 Classification: FATTY ACID BINDING PROTEIN/HYDROLASE |
Organism: Homo sapiens, Enterobacteria phage t4
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
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Gpr40 In Complex With Agopam Ap8 And Partial Agonist Mk-8666
Organism: Homo sapiens, Enterobacteria phage t4
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2017-06-07 Classification: FATTY ACID BINDING PROTEIN/HYDROLASE Ligands: OLC, MK6, 7OS |
Organism: Homo sapiens, Enterobacteria phage t4
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: OLC, MK6, 7OS
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Selective Small Molecule Inhibition Of The Fmn Riboswitch
Organism: Fusobacterium nucleatum
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2015-10-07 Classification: RNA/INHIBITOR Ligands: K, MG, 51B |
Organism: Fusobacterium nucleatum
Method: X-RAY DIFFRACTION
Release Date: 2015-10-07
Ligands: K, MG, 51B
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Irak4-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2015-09-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4S1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-02
Ligands: 4S1
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Irak4-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2015-09-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4S2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-02
Ligands: 4S2
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Irak4-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2015-09-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4S3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-02
Ligands: 4S3
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Kinase Domain Of Csrc In Complex With A Hinge Region-Binding Fragment
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-04-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0UL |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2013-04-10
Ligands: 0UL
