Search Count: 16
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Crystal Structure Of Rar-Related Orphan Receptor C In Complex With A Novel Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-08-12 Classification: TRANSCRIPTION/Agonist Ligands: V27 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: V27
 |
Crystal Structure Of Rar-Related Orphan Receptor C In Complex With A Potent, Selective And Orally Bioavailable Ror-Gamma-T Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2020-08-12 Classification: TRANSCRIPTION/AGONIST Ligands: VBG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: VBG, SO4
 |
Structure Of Human Pregnane X Receptor Ligand Binding Domain Bound Tethered With Src Co-Activator Peptide And Compound-3 Aka 1,1,1,3,3,3-Hexafluoro-2-{4-[1-(4- Luorobenzenesulfonyl)Cyclopentyl]Phenyl}Propan-2-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2020-02-12 Classification: TRANSFERASE Ligands: L7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-12
Ligands: L7D
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Crystal Structure Of Rar-Related Orphan Receptor C In Complex With A Phenyl (3-Phenylpyrrolidin-3-Yl)Sulfone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2019-03-20 Classification: TRANSCRIPTION/INHIBITOR Ligands: L8A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-20
Ligands: L8A
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Identification Of Bicyclic Hexafluoroisopropyl Alcohol Sulfonamides As Rorgt/Rorc Inverse Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-12-20 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: XGH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: XGH, SO4
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Structure Of Human Pregnane X Receptor Ligand Binding Domain Bound Tethered With Src Co-Activator Peptide And Compound 25A Aka Bicyclic Hexafluoroisopropyl 2 Alcohol Sulfonamides
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2017-12-20 Classification: NUCLEAR PROTEIN Ligands: XGH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: XGH
 |
P38 Alpha Kinase Complexed With A Pyrazolo-Triazine Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2012-02-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: NK0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-01
Ligands: NK0
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P38 Alpha Kinase Complexed With A 5-Amino-Pyrazole Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2010-11-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OCG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-17
Ligands: OCG
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P38 Alpha Map Kinase Complexed With Pyrrolotriazine Inhibitor 7K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-10-13 Classification: TRANSFERASE Ligands: 38P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: 38P
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P38 Alpha Map Kinase Complexed With Pyrrolotriazine Inhibitor 7V
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-10-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 39P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: 39P
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P38 Alpha Kinase Complexed With A Pyrazolo-Pyrimidine Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2010-03-02 Classification: TRANSFERASE Ligands: N4D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: N4D
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Morpholino Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2008-04-15 Classification: TRANSFERASE Ligands: P39 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-15
Ligands: P39
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P38 Alpha Map Kinase Complexed With Bms-640994
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-04-15 Classification: SIGNALING PROTEIN, TRANSFERASE Ligands: 304 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-15
Ligands: 304
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Morpholino Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-04-08 Classification: TRANSFERASE Ligands: P38 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-08
Ligands: P38
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Phenylalanine Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 11B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: 279 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: 279
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Phenylalanine Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 11J
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: 287 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: 287