Search Count: 13
![]() |
Pqr530 [(S)-4-(Difluoromethyl)-5-(4-(3-Methylmorpholino)-6-Morpholino-1,3,5-Triazin-2-Yl)Pyridin-2-Amine] Bound To The Pi3Ka Catalytic Subunit P110Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2019-06-26 Classification: TRANSFERASE Ligands: M1J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: M1J
![]() |
Pqr309 - A Potent, Brain-Penetrant, Orally Bioavailable, Pan-Class I Pi3K/Mtor Inhibitor As Clinical Candidate In Oncology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-09-06 Classification: TRANSFERASE Ligands: A3W, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-06
Ligands: A3W, SO4
![]() |
Complex Between The Leucine Zipper (Lz) And Centrosomin-Motif 2 (Cm2) Domains Of Drosophila Melanogaster Centrosomin (Cnn)
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2017-06-28 Classification: CELL CYCLE Ligands: ZN, CL, EDO |
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: ZN, CL, EDO
![]() |
Complex Between The Leucine Zipper (Lz) And Centrosomin-Motif 2 (Cm2) Domains Of Drosophila Melanogaster Centrosomin (Cnn) - L535E Mutant Form
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-06-28 Classification: CELL CYCLE Ligands: ZN |
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: ZN
![]() |
Complex Between The Leucine Zipper (Lz) And Centrosomin-Motif 2 (Cm2) Domains Of Drosophila Melanogaster Centrosomin (Cnn) - L535E Mutant Form
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-06-28 Classification: CELL CYCLE Ligands: ZN |
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: ZN
![]() |
Complex Between The Leucine Zipper (Lz, Residues 490-567) And Centrosomin-Motif 2 (Cm2) Domains Of Drosophila Melanogaster Centrosomin (Cnn)
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2017-06-28 Classification: CELL CYCLE Ligands: ZN, EDO, TCE |
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: ZN, EDO, TCE
![]() |
Tubulin Mtd265-R1 Complex
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-03-22 Classification: CELL CYCLE Ligands: GTP, MG, CA, GOL, UGI, GDP, MES, ACP |
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-03-22
Ligands: GTP, MG, CA, GOL, UGI, GDP, MES, ACP
![]() |
Structure Of Phosphoinositide 3-Kinase Gamma (Pi3K) Bound To The Potent Inhibitor Pikin2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2017-03-15 Classification: TRANSFERASE Ligands: 6K7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 6K7, SO4
![]() |
Structure Of Phosphoinositide 3-Kinase Gamma (Pi3K) Bound To The Potent Inhibitor Pikin3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2017-03-15 Classification: TRANSFERASE Ligands: 6K5, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 6K5, SO4
![]() |
Centrosomin-Motif 2 (Cm2) Domain Of Drosophila Melanogaster Centrosomin (Cnn)
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-03-08 Classification: STRUCTURAL PROTEIN Ligands: ZN |
Organism: Drosophila melanogaster
Method: X-RAY DIFFRACTION
Release Date: 2017-03-08
Ligands: ZN
![]() |
Tubulin-Bkm120 Complex
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2017-02-22 Classification: CELL CYCLE Ligands: GTP, MG, CA, GOL, GDP, MES, SD5, ACP |
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: GTP, MG, CA, GOL, GDP, MES, SD5, ACP
![]() |
Tubulin-Mtd147 Complex
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-02-22 Classification: CELL CYCLE Ligands: GTP, MG, CA, GOL, FB7, GDP, MES, ACP |
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: GTP, MG, CA, GOL, FB7, GDP, MES, ACP
![]() |
Tubulin-Mtd265 Complex
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2017-02-22 Classification: CELL CYCLE Ligands: GTP, MG, CA, GOL, 918, GDP, MES, ACP |
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: GTP, MG, CA, GOL, 918, GDP, MES, ACP
