Search Count: 16
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Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 2-(3-(1-(4-Chlorophenyl)Cyclopropyl) -[1,2,4]Triazolo[4,3-A]Pyridin-8-Yl)Propan-2-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2018-12-19 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, HJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: NAP, HJG
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Crystal Structure Of Murine 11B- Hydroxysteroiddehydrogenase Complexed With 2-(3-(1-(4- Chlorophenyl)Cyclopropyl)-[1,2,4]Triazolo[4,3-A]Pyridin-8- Yl)Propan-2-Ol
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2018-12-19 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, HJG, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: NAP, HJG, SO4
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Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 2-[2-(4-Fluorophenyl)-2-Adamantyl]-1-(3-Methoxyazetidin-1-Yl)Ethanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8K4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8K4
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Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 1-(3-Hydroxyazetidin-1-Yl)-2-[(2S,5R)-2-(4-Fluorophenyl)-5-Methoxyadamantan-2-Yl]Ethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8K7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8K7
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Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 2-[(1R,3S,5R,7S)-2-[4-(4-Fluorophenyl)Phenyl]-6-Hydroxyadamantan-2-Yl]-1-(3- Hydroxyazetidin-1-Yl)Ethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8KA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8KA
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Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 2-(2-Benzyl-6-Hydroxyadamantan-2-Yl)-1-(3-Hydroxyazetidin-1-Yl)Ethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8KD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8KD
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Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 2-[(5R,7S)-6-Hydroxy-2-Phenyladamantan-2-Yl]-1-(3-Hydroxyazetidin-1-Yl)Ethan-1-One (Bms-816336)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8KG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8KG
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Crystal Structure Of Murine 11Beta- Hydroxysteroiddehydrogenase Complexed With 2-[(5R,7S)-6-Hydroxy-2-Phenyladamantan-2-Yl]-1-(3-Hydroxyazetidin-1-Yl)Ethan-1-One (Bms-816336)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8KG, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8KG, SO4
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Crystal Structure Of 11B-Hsd1 Double Mutant (L262R, F278E) In Complex With (1S,4S)-4-[8-(2-Fluorophenoxy)[1,2,4]Triazolo[4,3-A]Pyridin-3-Yl]Bicyclo[2.2.1]Heptan-1-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2014-06-11 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 1EO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: NAP, 1EO, CL
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Crystal Structure Of 11B-Hsd1 Double Mutant (L262R, F278E) In Complex With 3-[1-(4-Chlorophenyl)Cyclopropyl]-8-(2-Fluorophenoxy)[1,2,4]Triazolo[4,3-A]Pyridine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2014-06-11 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 1EN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: NAP, 1EN
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Crystal Structure Of 11B-Hsd1 Double Mutant (L262R, F278E) In Complex With 3-[1-(4-Chlorophenyl)Cyclopropyl]-8-Cyclopropyl[1,2,4]Triazolo[4,3-A]Pyridine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2014-06-11 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 1EQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: NAP, 1EQ
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Crystal Structure Of 11B-Hsd1 Double Mutant (L262R, F278E) Complexed With 8-{[(2-Cyanopyridin-3-Yl)Methyl]Sulfanyl}-6-Hydroxy-3,4-Dihydro-1H-Pyrano[3,4-C]Pyridine-5-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-11-02 Classification: Oxidoreductase/Oxidoreductase Inhibitor Ligands: NAP, 07M, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-02
Ligands: NAP, 07M, GOL
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Crystal Structure Of The Rat Androgen Receptor Ligand Binding Domain Complex With An N-Aryl-Oxazolidin 2-Imine Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2009-04-28 Classification: HORMONE Ligands: LGB |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2009-04-28
Ligands: LGB
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Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With (3,3-Dimethylpiperidin-1-Yl)(6-(3-Fluoro-4-Methylphenyl)Pyridin-2-Yl)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2008-06-10 Classification: OXIDOREDUCTASE Ligands: NAP, 311 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-10
Ligands: NAP, 311
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Crystal Structure Of The Rat Androgen Receptor Ligand Binding Domian Complex With An N-Aryl-Hydroxybicyclohydantoin
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2006-12-12 Classification: HORMONE/GROWTH FACTOR Ligands: LG7 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2006-12-12
Ligands: LG7
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Crystal Structure Of The Rat Androgen Receptor Ligand Binding Domain Complex With Bms-564929
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2006-12-12 Classification: HORMONE/GROWTH FACTOR Ligands: 8NH |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2006-12-12
Ligands: 8NH