Search Count: 27
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Inhibitor Bound Vim1
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2024-10-16 Classification: HYDROLASE Ligands: MG, ZN, A1AUQ |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: MG, ZN, A1AUQ
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Inhibitor Bound Vim1
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.01 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: ZN, OKC |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: ZN, OKC
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Inhibitor Bound Vim1
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: ZN, OK0 |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: ZN, OK0
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Inhibitor Bound Vim1
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.02 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: MG, ZN, OJR |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: MG, ZN, OJR
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Inhibitor Bound Vim1
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.00 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: EDO, ACT, ZN |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: EDO, ACT, ZN
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Structure Of Lrrk2-Chk1 10-Pt. Mutant Complex With Heteroaryl-1H-Indazole Lrrk2 Inhibitor 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2023-02-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: UUF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-22
Ligands: UUF
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Structure Of Lrrk2-Chk1 10-Pt. Mutant Complex With Heteroaryl-1H-Indazole Lrrk2 Inhibitor 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2023-02-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: UU6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-22
Ligands: UU6
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Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2021-06-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-16
Ligands: YXD
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Crystal Structure Of The Spa17 Docking And Dimerization Domain From Danio Rerio
Organism: Danio rerio
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2021-05-26 Classification: PROTEIN BINDING |
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
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Discovery Of Mli-2, An Orally Available And Selective Lrrk2 Inhibitor That Reduces Brain Kinase Activity
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2017-03-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 81Y, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 81Y, SO4
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Bace1 In Complex With (S)-5-(3-Chloro-5-(5-(Prop-1-Yn-1-Yl)Pyridin-3-Yl)Thiophen-2-Yl)-2,5-Dimethyl-1,2,4-Thiadiazinan-3-Iminium 1,1-Dioxide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 66J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 66J
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Bace1 In Complex With 4-(3-(Furan-2-Carboxamido)Phenyl)-1-Methyl-5-Oxo-4-Phenylimidazolidin-2-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: TLA, 66H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: TLA, 66H
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Bace1 In Complex With (R)-N-(3-(3-Amino-2,5-Dimethyl-1,1-Dioxido-5,6-Dihydro-2H-1,2,4-Thiadiazin-5-Yl)-4-Fluorophenyl)-5-Fluoropicolinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 66F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 66F
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Crystal Structure Of The Central Domain Of Human Akap18 Gamma/Delta In Complex With Malonate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2016-08-03 Classification: HYDROLASE Ligands: MLI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-03
Ligands: MLI
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Structure Of Shigella Effector Ospg In Complex With Host Ubch5C- Ubiquitin Conjugate
Organism: Shigella flexneri, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2014-01-29 Classification: TRANSFERASE/LIGASE/PROTEIN BINDING |
Organism: Shigella flexneri, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-29
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Pseudo-Atomic Model Of The Akap18-Pka Complex In A Bent Conformation Derived From Electron Microscopy
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY Release Date: 2013-11-13 Classification: TRANSFERASE |
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY
Release Date: 2013-11-13
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Pseudo-Atomic Model Of The Akap18-Pka Complex In A Linear Conformation Derived From Electron Microscopy
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY Release Date: 2013-11-13 Classification: TRANSFERASE |
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY
Release Date: 2013-11-13
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Structure Of Bace In Complex With (S)-4-(3-Chloro-5-(5-(Prop-1-Yn-1-Yl)Pyridin-3-Yl)Thiophen-2-Yl)-1,4-Dimethyl-6-Oxotetrahydropyrimidin-2(1H)-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-08-08 Classification: Hydrolase/Hydrolase inhibitor Ligands: 0V6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: 0V6
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Akap18 Delta Central Domain - Amp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2008-05-06 Classification: HYDROLASE Ligands: AMP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-05-06
Ligands: AMP
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Akap18 Delta Central Domain - Cmp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2008-05-06 Classification: HYDROLASE Ligands: C5P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-05-06
Ligands: C5P
