Search Count: 20
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Cobimetinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2020-10-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, EUI |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-10-07
Ligands: ANP, MG, EUI
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Crystal Structure Of Ksr2:Mek1 In Complex With Adp
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ADP, MG |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ADP, MG
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Trametinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, QOM |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, QOM
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Cobimetinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, VKD |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, VKD
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Crystal Structure Of Ksr2:Mek1 In Complex With Anp-Pnp, And Allosteric Mek Inhibitor Selumetinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.09 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, 3EW |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, 3EW
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Pd0325901
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.19 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, 4BM |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, 4BM
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Aps-9-95-1
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.36 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, VKG |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, VKG
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Trametinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.34 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, QOM |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, QOM
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Selumetinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.21 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, 3EW |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, 3EW
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Pd0325901
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.63 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, 4BM |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, 4BM
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Aps-9-95-1
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.62 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, VKG |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, VKG
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Ksr2:Mek1 Complex Bound To The Small Molecule Aps-2-79
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.51 Å Release Date: 2016-08-31 Classification: TRANSFERASE Ligands: 6U7 |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 6U7
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Crystal Structure Of Human Dot1L In Complex With Inhibitor Epz004777
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-05-16 Classification: Transferase/Transferase Inhibitor Ligands: 0QK, SO4, EDO, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: 0QK, SO4, EDO, UNX
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Crystal Structure Of Human Dot1L In Complex With 2 Molecules Of Epz004777
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2012-05-16 Classification: Transferase/Transferase Inhibitor Ligands: 0QK, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: 0QK, UNX
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Crystal Structure Of Human Dot1L In Complex With Inhibitor Sgc0946
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2012-05-16 Classification: Transferase/Transferase Inhibitor Ligands: BR, AW2, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: BR, AW2, NA
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Crystal Structure Of Human Dot1L In Complex With Inhibitor Sgc0947
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-05-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: AW3, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: AW3, GOL
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Crystal Structure Of Human Dot1L In Complex With Inhibitor Fed2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2012-05-02 Classification: Transferase/Transferase Inhibitor Ligands: AW0, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-02
Ligands: AW0, UNX
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Crystal Structure Of Human Dot1L In Complex With Inhibitor Fed1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-05-02 Classification: Transferase/Transferase Inhibitor Ligands: AW1, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-02
Ligands: AW1, UNX
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Crystal Structure Of Dot1L In Complex With 5-Iodotubercidin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2012-03-14 Classification: TRANSFERASE Ligands: 5ID, IOD, NA, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-14
Ligands: 5ID, IOD, NA, UNX