Search Count: 19
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Crystal Structure Of The Peptidoglycan O-Acetyltransferase B (Patb) From Campylobacter Jejuni, Catalytic Domain
Organism: Campylobacter jejuni
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: CL |
Organism: Campylobacter jejuni
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: CL
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Crystal Structure Of Hiv-1 Protease With Gs-9770
Organism: Hiv-1 06tg.ht043
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2024-03-06 Classification: VIRAL PROTEIN Ligands: A1AAD |
Organism: Hiv-1 06tg.ht043
Method: X-RAY DIFFRACTION
Release Date: 2024-03-06
Ligands: A1AAD
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Mth1 In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2020-04-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: S3O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: S3O
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Mth1 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2020-04-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 8JF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: 8JF
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Mth1 In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-04-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GN6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: GN6
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Crystal Structure Of Hcv Ns3/4A Protease In Complex With Voxilaprevir
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2019-07-10 Classification: viral protein/inhibitor Ligands: L9P, ZN, SO4 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: L9P, ZN, SO4
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Crystal Structure Of Hcv Ns3/4A Protease In Complex With Compound 12
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2019-07-10 Classification: viral protein/inhibitor Ligands: L9J, ZN, SO4 |
Organism: Hepatitis c virus subtype 1a
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: L9J, ZN, SO4
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Ask1 Kinase Domain Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-09-19 Classification: TRANSFERASE/INHIBITOR Ligands: KK7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: KK7
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Ask1 Kinase Domain Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-09-19 Classification: TRANSFERASE/INHIBITOR Ligands: KK8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: KK8
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Ask1 Kinase Domain Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2018-09-19 Classification: TRANSFERASE/INHIBITOR Ligands: S0L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: S0L
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Structure Determination Of A Potent, Selective Antibody Inhibitor Of Human Mmp9 (Gs-5745 Bound To Mmp-9)
Organism: Oryctolagus cuniculus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2017-03-15 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA, NCO |
Organism: Oryctolagus cuniculus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: ZN, CA, NCO
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Structure Determination Of A Potent, Selective Antibody Inhibitor Of Human Mmp9 (Apo Mmp9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2017-03-01 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: ZN, CA
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 3) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 7HG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 7HG
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 5) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78E
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 6) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78R
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 7) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78X
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 8) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 838, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 838, SO4
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Idelalisib Bound To The P110 Subunit Of Pi3K Delta
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2015-02-04 Classification: Transferase/transferase inhibitor Ligands: 40L |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 40L
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Discovery Of A Novel Hydroxy Pyrazole Based Factor Ixa Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2006-04-04 Classification: HYDROLASE/BLOOD CLOTTING Ligands: 6NH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-04-04
Ligands: 6NH
