Search Count: 22
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Cryo-Em Structure Of Ccr6 Bound By Pf-07054894 And Oxm2
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY Resolution:3.35 Å Release Date: 2025-10-01 Classification: MEMBRANE PROTEIN Ligands: A1A1W, A1CH1 |
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2025-10-01
Ligands: A1A1W, A1CH1
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Pad2 With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2025-07-30 Classification: HYDROLASE Ligands: A1CE0, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-30
Ligands: A1CE0, CA
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2025-05-28 Classification: HYDROLASE Ligands: CA, A1A8O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1A8O
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Inhibiting Peptidylarginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, A1BZK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1BZK
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1A9P, 3YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1A9P, 3YZ
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Cryo-Em Structure Of Ccr6 Bound By Sqa1 And Oxm2
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY Release Date: 2024-09-11 Classification: MEMBRANE PROTEIN Ligands: CLR, EBX, A1A1W |
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2024-09-11
Ligands: CLR, EBX, A1A1W
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Cryo-Em Structure Of Ccr6 Bound By Sqa1 And Oxm1
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY Release Date: 2024-09-11 Classification: MEMBRANE PROTEIN Ligands: CLR, EBX, A1A2A |
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2024-09-11
Ligands: CLR, EBX, A1A2A
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Human Retenoid-Related Orphan Receptor-Gamma (Rorc2) Ligand-Binding Domain In Complex With Compound 5 Andindazole Acid Bound In H12-Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-03-01 Classification: DNA BINDING PROTEIN Ligands: LKY, 4Y5, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: LKY, 4Y5, SO4
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Human Retenoid-Related Orphan Receptor-Gamma (Rorc2) Ligand-Binding Domain In Complex With Compound 6A Andindazole Acid Bound In H12-Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2023-03-01 Classification: DNA BINDING PROTEIN Ligands: XNR, 4Y5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: XNR, 4Y5
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Human Retenoid-Related Orphan Receptor-Gamma (Rorc2) Ligand-Binding Domain In Complex With Compound 8 Andindazole Acid Bound In H12-Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-03-01 Classification: DNA BINDING PROTEIN Ligands: XO5, XNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: XO5, XNX
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Crystal Structure Of Mouse Btk Kinase Domain In Complex With Compound 9A
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-01-30 Classification: TRANSFERASE Ligands: JVP |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-01-30
Ligands: JVP
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Human Retenoid-Related Orphan Receptor-Gamma Ligand- Binding Domain In Complex With Indole Ligand Cp9B In Inverse Agonist Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-09-05 Classification: SIGNALING PROTEIN Ligands: F7M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: F7M
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Rorc2 Lbd Complexed With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2018-09-05 Classification: SIGNALING PROTEIN Ligands: F7J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: F7J
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Crystal Structure Of Btk Mutant (F435T,K596R) Complexed With Imidazo[1,5-A]Quinoxaline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2011-10-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: IAQ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: IAQ, GOL
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Crystal Structure Of Human Mmp-13 Complexed With An Amino-2-Indanol Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-02-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, ZN, SO4, LA3, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: CA, ZN, SO4, LA3, EPE
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Crystal Structure Of Human Mmp-13 Complexed With A Phenyl-2H-Tetrazole Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2010-11-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, 3KE, HAE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: ZN, CA, SO4, 3KE, HAE
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Crystal Structure Of Human Mmp-13 Complexed With A (Pyridin-4-Yl)-2H-Tetrazole Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2010-11-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, 3EJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: ZN, CA, 3EJ
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Crystal Structure Of Human Mmp-13 Complexed With A (Pyridin-4-Yl)-2H-Tetrazole Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2010-11-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, 3EK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: ZN, CA, 3EK
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Crystal Structure Of The Catalytic Domain Of Adamts-5 In Complex With An Amino-2-Indanol Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2010-03-31 Classification: HYDROLASE Ligands: LA3, EDO, ZN, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-31
Ligands: LA3, EDO, ZN, CA
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Crystal Structure Of The Catalytic Domain Of Adamts-5 In Complex With Marimastat
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2009-07-07 Classification: HYDROLASE Ligands: 097, ZN, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-07
Ligands: 097, ZN, CA
