Search Count: 24
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Ternary Complex Of Crbn-Ddb1-Ppil4 Rrm Domain With Fpft-2216
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-08-06 Classification: LIGASE Ligands: ZN, A1BC8 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-08-06
Ligands: ZN, A1BC8
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Ternary Complex Of Crbn-Ddb1-Pde6D With Fpft-2216
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-08-06 Classification: LIGASE Ligands: ZN, A1BC8 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-08-06
Ligands: ZN, A1BC8
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Cryo-Em Structure Of Ddb1Deltab-Dda1-Dcaf5
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-03
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Egfr (T79M/V948R) In Complex With Naquotinib And An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2022-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: VNS, 8RC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: VNS, 8RC
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Egfr L858R/V948R In Complex With Osimertinib And Allosteric Inhibitor Jbj-09-063
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2021-09-15 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: VNS, YY3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VNS, YY3
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Egfr Kinase (L858R/V948R) In Complex With Allosteric Inhibitor Jbj-09-063
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2021-09-15 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: MG, ANP, VNS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: MG, ANP, VNS
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Egfr Kinase (T790M/V948R) In Complex With Pf-06747775
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: 8BS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: 8BS
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Egfr Kinase (T790M/V948R) In Complex With Pf-06747775 And Jbj-04-125-02
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ANP, MG, JBJ, 8BS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ANP, MG, JBJ, 8BS
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Egfr Kinase (T790M/V948R) In Complex With Az5104
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: VO7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: VO7
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Egfr Kinase (T790M/V948R) In Complex With Osimertinib And Eai045
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ANP, MG, 9LL, YY3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ANP, MG, 9LL, YY3
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Egfr Kinase (T790M/V948R) In Complex With Osimertinib And Jbj-04-125-02
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ANP, MG, JBJ, YY3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ANP, MG, JBJ, YY3
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Egfr Kinase (T790M/V948R) In Complex With Osimertinib And Jbj-09-063
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: YY3, VNS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: YY3, VNS
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Egfr(T790M/V948R) In Complex With Azd9291 And Ddc4002
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2021-06-30 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: Q6K, NQ1, MG, ANP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-30
Ligands: Q6K, NQ1, MG, ANP
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Egfr(T790M/V948R) In Complex With Ln3844
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2021-05-19 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: UEJ, ANP, MG, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: UEJ, ANP, MG, CL
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Crystal Structure Of The Braf:Mek1 Kinases In Complex With Amppnp And Selumetinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.19 Å Release Date: 2021-04-21 Classification: TRANSFERASE Ligands: 3EW, ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: 3EW, ANP, MG
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Crystal Structure Of The Braf:Mek1 Kinases In Complex With Amppnp And Binimetinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.09 Å Release Date: 2021-04-21 Classification: TRANSFERASE Ligands: ANP, MG, QO7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: ANP, MG, QO7
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Crystal Structure Of The Braf:Mek1 Kinases In Complex With Amppnp And Cobimetinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.16 Å Release Date: 2021-04-21 Classification: TRANSFERASE Ligands: ANP, MG, EUI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: ANP, MG, EUI
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Crystal Structure Of The Braf:Mek1 Kinases In Complex With Amppnp And Pimasertib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.09 Å Release Date: 2021-04-21 Classification: TRANSFERASE Ligands: ANP, MG, QOA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: ANP, MG, QOA
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Crystal Structure Of The Braf:Mek1 Kinases In Complex With Amppnp And Pd0325901
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2021-04-21 Classification: TRANSFERASE Ligands: ANP, MG, CL, 4BM, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: ANP, MG, CL, 4BM, SO4, GOL
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Crystal Structure Of The Braf:Mek1 Kinases In Complex With Amppnp And Trametinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.45 Å Release Date: 2021-04-21 Classification: TRANSFERASE Ligands: ANP, MG, SO4, QOM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: ANP, MG, SO4, QOM
