Search Count: 14
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Tead1 In Complex With A Reversible Inhibitor N-[(1S)-2-Hydroxy-1-(1-Methyl-1H-Pyrazol-3-Yl)Ethyl]-2-Methyl-8-[4-(Trifluoromethyl)Phenyl]-2H,8H-Pyrazolo[3,4-B]Indole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2025-01-22 Classification: TRANSCRIPTION Ligands: GOL, A1IJL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: GOL, A1IJL, SO4
 |
Tead1/Yap In Complex With A Reversible Inhibitor N-[(4-Phenoxyphenyl)Methyl]Imidazo[1,2-A]Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2024-10-16 Classification: TRANSCRIPTION Ligands: CL, A1IHH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: CL, A1IHH
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Vcb In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2023-02-15 Classification: LIGASE Ligands: QF7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
Ligands: QF7
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Vcb In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2023-02-15 Classification: LIGASE Ligands: QE0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
Ligands: QE0
 |
Vcb In Complex With Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-02-15 Classification: LIGASE Ligands: QF3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
Ligands: QF3
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Vcb In Complex With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2023-02-15 Classification: LIGASE Ligands: QE9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
Ligands: QE9
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Vcb In Complex With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2023-02-15 Classification: LIGASE Ligands: QFR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
Ligands: QFR
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Vcb In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2023-02-15 Classification: LIGASE Ligands: QFF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
Ligands: QFF
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Ternary Complex Between Vcb, Brd4-Bd1 And Protac 48
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2023-02-15 Classification: LIGASE Ligands: SO4, EDO, QIY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
Ligands: SO4, EDO, QIY
 |
Ternary Complex Between Vcb, Brd4-Bd2 And Protac 51
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2023-02-15 Classification: LIGASE Ligands: QLX, MLI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
Ligands: QLX, MLI
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Ternary Complex Between Vcb, Brd4-Bd2 And Protac 48
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2023-02-15 Classification: LIGASE Ligands: QIY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
Ligands: QIY
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Ternary Complex Between Vcb, Brd4-Bd1 And Protac 49
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.18 Å Release Date: 2023-02-15 Classification: LIGASE Ligands: SO4, QIK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
Ligands: SO4, QIK
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Optimization Of Tead P-Site Binding Fragment Hit Into In Vivo Active Lead Msc-4106
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JJU, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: JJU, SO4
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Human Tead3 In Complex With 1-Cyclopentyl-1H-Pyrazolo[3,4-B]Pyridine-5-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JIK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: JIK