Search Count: 103
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Crystal Structure Of The Smarca2 Bromodomain Bound To A Fragment Screening Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2025-06-18 Classification: GENE REGULATION Ligands: A1I5P, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-18
Ligands: A1I5P, ZN
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Pyrazine Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2025-05-28 Classification: TRANSFERASE Ligands: A1JAF, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1JAF, EDO
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Crystal Structure Of The Smarca2 Bromodomain Bound To A Tricyclic Pyrimidoindolone Inhibitor (Compound 17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2025-05-14 Classification: GENE REGULATION Ligands: A1I45, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1I45, ZN
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITC
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITA
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Pyrazine Carboxamide Inhibitor Az3246 (Compound 24)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITB, EDO
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Crystal Structure Of Human Cdc20 Bound To Synthetic D-Box Peptide D21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2025-02-12 Classification: LIGASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
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Crystal Structure Of Human Cdc20 Bound To Synthetic D-Box Peptide D20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2025-02-12 Classification: LIGASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
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Crystal Structure Of Human Cdc20 Bound To Synthetic D-Box Peptide D7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2025-02-12 Classification: LIGASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
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E3 Ligase Cbl-B In Complex With A Triazolone Core Inhibitor (Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IEW, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IEW, ZN, NA
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E3 Ligase Cbl-B In Complex With A Lactam Scaffold Inhibitor (Compound 7)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IEV, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IEV, ZN, NA
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E3 Ligase Cbl-B In Complex With A Carbamate Scaffold Inhibitor (Compound 12)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IE5, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IE5, ZN, NA
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Crystal Structure Of Human Ampk Heterotrimer In Complex With Allosteric Activator C455
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2024-05-15 Classification: SIGNALING PROTEIN Ligands: STU, QTN, AMP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-15
Ligands: STU, QTN, AMP
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Crystal Structure Of Human Mat2A Bound To S-Adenosylmethionine And Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2024-03-20 Classification: TRANSFERASE Ligands: U74, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: U74, SAM
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Crystal Structure Of Human Mat2A Bound To S-Adenosylmethionine And Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2024-03-20 Classification: TRANSFERASE Ligands: U6R, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: U6R, SAM
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Crystal Structure Of Human Mat2A Bound To S-Adenosylmethionine And Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2024-03-20 Classification: TRANSFERASE Ligands: U8R, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: U8R, SAM
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Crystal Structure Of Human Mat2A Bound To S-Adenosylmethionine And Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2024-03-20 Classification: TRANSFERASE Ligands: U8E, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: U8E, SAM
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Crystal Structure Of Human Mat2A Bound To S-Adenosylmethionine And Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2024-03-20 Classification: TRANSFERASE Ligands: U7X, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: U7X, SAM