Search Count: 16
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Egfr(T790M/V948R) In Complex With Ln5461
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2024-08-28 Classification: TRANSFERASE Ligands: MG, ANP, IXC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-08-28
Ligands: MG, ANP, IXC
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Egfr(T790M/V948R) In Complex With The Allosteric Inhibitor Frf-06-057
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2024-08-28 Classification: TRANSFERASE Ligands: MG, ANP, IXR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-08-28
Ligands: MG, ANP, IXR
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Egfr(T790M/V948R) In Complex With Compound 1 (Ln4503)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-01-17 Classification: TRANSFERASE Ligands: MG, ANP, YA6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-17
Ligands: MG, ANP, YA6
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Egfr(T790M/V948R) In Complex With Compound 2 (Ln5993)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2024-01-17 Classification: TRANSFERASE Ligands: YAA, MG, ANP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-17
Ligands: YAA, MG, ANP
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Egfr Kinase In Complex With Tas6417 (Cln-081)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2023-11-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: X9H, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: X9H, CIT
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Egfr(T790M/V948R) Kinase In Complex With Poziotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2023-11-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R2E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: R2E
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Egfr Kinase In Complex With Mobocertinib (Tak-788)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-11-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R28 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: R28
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Egfr Kinase In Complex With Poziotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2023-11-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R2E, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: R2E, CIT
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Egfr Kinase In Complex With Bayer #33
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-11-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: X9B, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: X9B, CIT
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Egfr(T790M/V948R) In Complex With A Macrocyclic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.42 Å Release Date: 2022-11-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M1O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: M1O
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Egfr Kinase In Complex With A Macrocyclic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-11-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0R, FLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: M0R, FLC
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Egfr In Complex With A Macrocyclic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2022-11-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M19, FLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: M19, FLC
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Wild Type Egfr In Complex With Lazertinib (Yh25448)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2022-11-23 Classification: TRANSFERASE/INHIBITOR Ligands: ZRT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: ZRT
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Egfr(T790M/V948R) In Complex With Lazertinib (Yh25448)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2022-11-23 Classification: TRANSFERASE Ligands: ZRT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: ZRT
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Active Conformation Of Egfr Kinase In Complex With Bi-4020
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2022-01-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, XA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: CL, XA4
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Inactive Conformation Of Egfr (T790M/V948R) Kinase In Complex With Bi-4020
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2022-01-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: XA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: XA4
