Search Count: 19
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Crystal Structure Of Human Kras G12C Covalently Bound To A Phthalazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, OJ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: MG, GDP, OJ1
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Crystal Structure Of Human Kras G12C Covalently Bound To A Quinazolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: GDP, CA, OHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: GDP, CA, OHY
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Crystal Structure Of Human Kras G12C Covalently Bound To Amg 510
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-11-06 Classification: SIGNALING PROTEIN Ligands: MG, GDP, MOV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: MG, GDP, MOV
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O67 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O67
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O5V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O5V
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, O5Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: MG, GDP, O5Y
 |
Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O5S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O5S
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Crystal Structure Of Human Pi3K-Gamma In Complex With Quinoline-Containing Inhibitor 5G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-06-21 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 6RF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: SO4, 6RF
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Crystal Structure Of Gdp-Mannose 4,6 Dehydratase Bound To A Gdp-Fucose Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-08-17 Classification: LYASE/INHIBITOR Ligands: NAP, GDP, 6CK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-17
Ligands: NAP, GDP, 6CK
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Crystal Structure Of Gdp-Mannose 4,6 Dehydratase In Complex With Natural Inhibitor Gdp-Fucose
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-08-17 Classification: LYASE/INHIBITOR Ligands: NAP, GDP, GFB, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-17
Ligands: NAP, GDP, GFB, GOL
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Crystal Structure Of Human Pi3K-Gamma In Complex With Benzimidazole Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-12-30 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 5MT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: SO4, 5MT
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Crystal Structure Of Human Pi3K-Gamma In Complex With (S)-N-(1-(7-Fluoro-2-(Pyridin-2-Yl)Quinolin-3-Yl)Ethyl)-9H-Purin-6-Amine Amg319 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VC
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Crystal Structure Of Human Pi3K-Gamma In Complex With Phenylquinoline Inhibitor N-{(1S)-1-[8-Chloro-2-(3-Fluorophenyl)Quinolin-3-Yl]Ethyl}-9H-Purin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VD
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Crystal Structure Of Human Pi3K-Gamma In Complex With Pyridinylquinoline Inhibitor N-{(1S)-1-[8-Chloro-2-(2-Methylpyridin-3-Yl)Quinolin-3-Yl]Ethyl}-9H-Purin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VE, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VE, GOL
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Crystal Structure Of Bace1 In Complex With Hydroxyethylamine Inhibitor 37
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0K9, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: 0K9, GOL
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Structure Of Bace-1 (Beta-Secretase) In Complex With (2R)-N-((2S,3R)-1-(Benzo[D][1,3]Dioxol-5-Yl)-3-Hydroxy-4-((S)-6'-Neopentyl-3',4'-Dihydrospiro[Cyclobutane-1,2'-Pyrano[2,3-B]Pyridine]-4'-Ylamino)Butan-2-Yl)-2-Methoxypropanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-04-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: IOD, GOL, 0KN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-18
Ligands: IOD, GOL, 0KN
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Crystal Structure Of Pi3K-Gamma In Complex With A Quinoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2011-06-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 2NQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-08
Ligands: SO4, 2NQ
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Crystal Structure Of Pi3K-Gamma In Complex With Benzothiazole 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QJZ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: QJZ, SO4
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Crystal Structure Of Pi3K-Gamma In Complex With Benzothiazole 82
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, QK0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SO4, QK0