Search Count: 55
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Crystal Structure Of Pi3K-Alpha In Complex With Taselisib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: 799 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: 799
 |
Crystal Structure Of Pi3K-Alpha In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3W
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3R
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3N
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Gdc-9545 In Complex With Estrogen Receptor Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2021-06-02 Classification: TRANSCRIPTION Ligands: G9J, ZNM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-02
Ligands: G9J, ZNM
 |
Crystal Structure Of Bcl-Xl In Complex With Tetrahydroisoquinoline-Pyridine Based Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-10-21 Classification: APOPTOSIS/APOPTOSIS INHIBITOR Ligands: RQ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-21
Ligands: RQ7
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Crystal Structure Of Estrogen Receptor Alpha In Complex With Receptor Degrader 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2020-07-01 Classification: NUCLEAR PROTEIN Ligands: G9J, U6D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: G9J, U6D
 |
Crystal Structure Of Estrogen Receptor Alpha In Complex With Receptor Degrader 16Ab
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-02-20 Classification: NUCLEAR PROTEIN Ligands: G8Y, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G8Y, GOL
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Crystal Structure Of Estrogen Receptor Alpha In Complex With Receptor Degrader 16Aa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-02-20 Classification: NUCLEAR PROTEIN Ligands: G9J, NI, G91, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G9J, NI, G91, GOL
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Crystal Structure Of Arq 531 In Complex With The Kinase Domain Of Btk
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2018-09-05 Classification: SIGNALING PROTEIN/inhibitor Ligands: HRA, IMD, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: HRA, IMD, EDO
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N-Terminal Bromodomain Of Brd4 In Complex With Plx5981
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: EDO, 6JC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: EDO, 6JC
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N-Terminal Bromodomain Of Brd4 In Complex With Otx-015
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 6JE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: 6JE
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N-Terminal Bromodomain Of Brd4 In Complex With Otx-015
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: EDO, 6JF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: EDO, 6JF
 |
Crystal Structure Of Nicotinamide Phosphoribosyltransferase (Nampt) In Complex With Inhibitors 37
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-08-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6TA, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 6TA, PO4, EDO
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Lactate Dehydrogenase A In Complex With A Trisubstituted Piperidine-2,4-Dione Inhibitor Gne-140
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-18 Classification: Oxidoreductase/Oxidoreductase Inhibitor Ligands: NAD, SO4, GN0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: NAD, SO4, GN0
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P110Alpha/P85Alpha With Compound 5
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-01-27 Classification: Transferase/Transferase Inhibitor Ligands: 5H2 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H2
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P110Alpha With Gdc-0326
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2016-01-27 Classification: Transferase/Inhibitor Ligands: 5H5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H5, EDO
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P110Delta/P85Alpha With Gdc-0326
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2016-01-27 Classification: Transferase/Inhibitor Ligands: 5H5 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H5
 |
The Crystal Structure Of Human Nicotinamide Phosphoribosyltransferase (Nampt) In Complex With N-(4-{(S)-[1-(2-Methylpropyl)Piperidin-4-Yl]Sulfinyl}Benzyl)Furo[2,3-C]Pyridine-2-Carboxamide Inhibitor (Compound 21)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2015-02-11 Classification: Transferase/Transferase inhibitor Ligands: 3TQ, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3TQ, PO4, EDO
 |
The Crystal Structure Of Nampt In Complex With Gne-618
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2014-10-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2P1, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-22
Ligands: 2P1, PO4, EDO