Search Count: 13
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Ternary Complex Of Vhl/Brd4-Bd1/Compound9 (4-(3,5-Difluoropyridin-2-Yl)-N-(11-(((S)-1-((2S,4R)-4-Hydroxy-2-((4-(4-Methylthiazol-5-Yl)Benzyl)Carbamoyl)Pyrrolidin-1-Yl)-3,3-Dimethyl-1-Oxobutan-2-Yl)Amino)-11-Oxoundecyl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-02-24 Classification: PEPTIDE BINDING PROTEIN Ligands: WEP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-24
Ligands: WEP
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Brd4-Bd1 Compound6 (Methyl 4-(3,5-Difluoropyridin-2-Yl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxylate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2021-02-24 Classification: CELL CYCLE Ligands: WEM, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-24
Ligands: WEM, GOL
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Structure Of A Peptide-Based Photo-Affinity Cross-Linker With Herceptin Fc
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2019-01-16 Classification: IMMUNE SYSTEM |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
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Crystal Structure Of Pdk1 In Complex With Atp And The Pif-Pocket Ligand Rs1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, ATP, R1S, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: GOL, ATP, R1S, EPE
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Crystal Structure Of Pdk1 In Complex With Atp And The Pif-Pocket Ligand Rs2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, ATP, R2S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: GOL, ATP, R2S
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Crystal Structure Of Pdk1 In Complex With Atp And Piftide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ATP, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: ATP, GOL
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Crystal Structure Of Gackix L664C Tethered To 1-10
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-03-06 Classification: TRANSFERASE Ligands: KI1, EDO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: KI1, EDO
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Pdk1 Mutant Bound To Allosteric Disulfide Fragment Inhibitor 1F8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-03-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1F8, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-23
Ligands: 1F8, CL
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Pdk1 Mutant Bound To Allosteric Disulfide Fragment Activator 2A2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-03-23 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: 2A2, BI4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-23
Ligands: 2A2, BI4
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Pdk1 Mutant Bound To Allosteric Disulfide Fragment Activator Js30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-03-23 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: J30, BI4, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-23
Ligands: J30, BI4, SO4, CL
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Bim Bh3 Peptide In Complex With Bcl-Xl
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2009-03-10 Classification: APOPTOSIS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
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Alpha/Beta Foldamer In Complex With Bcl-Xl
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2009-03-10 Classification: APOPTOSIS Ligands: EDO |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
Ligands: EDO
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Biotin Carboxyl Carrier Domain Of Transcarboxylase (1.3S) [10-48] Deletion Mutant
Organism: Propionibacterium freudenreichii subsp. shermanii
Method: SOLUTION NMR Release Date: 2002-11-21 Classification: CARRIER PROTEIN |
Organism: Propionibacterium freudenreichii subsp. shermanii
Method: SOLUTION NMR
Release Date: 2002-11-21
