Search Count: 42
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Cdk6 To Cdk4 Active Site Surrogate In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2025-12-17 Classification: TRANSFERASE/INHIBITOR Ligands: A1CIF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-17
Ligands: A1CIF
 |
Cdk6 To Cdk4 Active Site Surrogate In Complex With Pf-07220060
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2025-12-17 Classification: TRANSFERASE/INHIBITOR Ligands: A1AZ4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-17
Ligands: A1AZ4
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Gsk3Beta In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2025-12-17 Classification: TRANSFERASE/INHIBITOR Ligands: A1CIF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-17
Ligands: A1CIF
 |
Crystal Structure Of Mastl Kinase Domain In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2025-01-22 Classification: TRANSFERASE/INHIBITOR Ligands: A1AAE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: A1AAE
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Crystal Structure Of Map4K4 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2025-01-22 Classification: TRANSFERASE/INHIBITOR Ligands: A1AAA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: A1AAA
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1E
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: SO4, A1A1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: SO4, A1A1D
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1C
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1B, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1B, CL
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1A
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-[6-Chloro-4-(9-Methyl-1-Oxa-4,9-Diazaspiro[5.5]Undec-4-Yl)-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl]Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2023-04-05 Classification: TRANSFERASE Ligands: XXF, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: XXF, SO4
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-{4-[(3R,5S)-3-Amino-5-Methylpiperidin-1-Yl]-6-Chloro-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl}Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3I
 |
Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-{4-[(2S,5R)-5-Amino-2-Methylpiperidin-1-Yl]-6-Chloro-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl}Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3O
 |
Pkceta Kinase Domain In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: XXF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: XXF
 |
Pkceta Kinase Domain In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3I
 |
Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-2-[(4-Methoxy-6-Methyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-7-[(R)-Methoxy(Oxetan-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2017-12-27 Classification: Transferase/Transferase Inhibitor Ligands: ZN, CJD |
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: ZN, CJD
 |
Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-7-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-2-[(4,6-Dimethyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2017-12-27 Classification: METAL BINDING PROTEIN Ligands: ZN, CJG |
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: ZN, CJG
 |
Crystal Structure Of The Egfr Kinase Domain (L858R, T790M, V948R) In Complex With A Covalent Inhibitor N-[(3R,4R)-4-Fluoro-1-{6-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]-9-(Propan-2-Yl)-9H-Purin-2-Yl}Pyrrolidin-3-Yl]Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2017-03-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8BP, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-22
Ligands: 8BP, SO4, GOL
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Crystal Structure Of The Egfr Kinase Domain (L858R, T790M, V948R) In Complex With A Covalent Inhibitor N-[(3R,4R)-4-Fluoro-1-{6-[(3-Methoxy-1-Methyl-1H-Pyrazol-4-Yl)Amino]-9-(Propan-2-Yl)-9H-Purin-2-Yl}Pyrrolidin-3-Yl]Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2017-03-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8AM, SO4, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-22
Ligands: 8AM, SO4, GOL, EDO
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Crystal Structure Of The Egfr Kinase Domain (L858R, T790M, V948R) In Complex With 4-(4-{[2-{[(3S)-1-Acetylpyrrolidin-3-Yl]Amino}-9-(Propan-2-Yl)-9H-Purin-6-Yl]Amino}Phenyl)-1-Methylpiperazin-1-Ium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2017-03-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8BM, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-22
Ligands: 8BM, SO4, GOL