Search Count: 35
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Nacht Domain Of Nlrp3 In Complex With Dfv890
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2025-03-19 Classification: IMMUNE SYSTEM Ligands: A1IUG, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-19
Ligands: A1IUG, ADP
 |
Structure Of Ddb1/Cdk12/Cyclin K With Molecular Glue Sr-4835
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.90 Å Release Date: 2024-10-16 Classification: TRANSCRIPTION Ligands: RMF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: RMF
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Crystal Structure Of Human Cdk12/Cyclin K In Complex With Inhibitor Sr-4835
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2023-11-22 Classification: TRANSCRIPTION Ligands: RMF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: RMF
 |
Sculpting A Uniquely Reactive Cysteine Residue For Site-Specific Antibody Conjugation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2022-06-08 Classification: IMMUNE SYSTEM Ligands: PEG, SO4, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-08
Ligands: PEG, SO4, MG
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Crystal Structure Of Casein Kinase 1 Delta (Ck1 Delta) Complexed With Sr3029 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2020-03-25 Classification: TRANSFERASE Ligands: EDO, K0E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-25
Ligands: EDO, K0E
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Crystal Structure Of Casein Kinase I Isoform Delta (Ck1 Delta) Complexed With Sr4133 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2020-03-25 Classification: TRANSFERASE Ligands: SO4, EDO, NA, K0B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-25
Ligands: SO4, EDO, NA, K0B
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Crystal Structure Of H38C2 K99R Mutation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-07-10 Classification: IMMUNE SYSTEM Ligands: FLC, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: FLC, SO4
 |
Structure Of Cathepsin B1 From Schistosoma Mansoni In Complex With Wrr391 Inhibitor
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2018-11-21 Classification: HYDROLASE Ligands: 9U8, ACT |
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION
Release Date: 2018-11-21
Ligands: 9U8, ACT
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Structure Of Cathepsin B1 From Schistosoma Mansoni In Complex With Wrr286 Inhibitor
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-11-21 Classification: HYDROLASE Ligands: VS4, ACT |
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION
Release Date: 2018-11-21
Ligands: VS4, ACT
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Matrix Metalloproteinase-13 Complexed With Selective Inhibitor Compound (S)-10A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2017-07-12 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA, 8OM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-12
Ligands: ZN, CA, 8OM
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Matrix Metalloproteinase-13 Complexed With Selective Inhibitor Compound (S)-17A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2017-07-12 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA, 8OJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-12
Ligands: ZN, CA, 8OJ
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Matrix Metalloproteinase-13 Complexed With Selective Inhibitor Compound (R)-17A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2017-07-12 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA, 8OA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-12
Ligands: ZN, CA, 8OA
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Matrix Metalloproteinase-13 Complexed With Selective Inhibitor Compound 10D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2017-07-12 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA, 8O7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-12
Ligands: ZN, CA, 8O7, SO4
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Crystal Structure Analysis Of Cruzain Bound To The No-Covalent Analog Of Wrr-483 (Wrr-669)
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2015-03-11 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 2VC, EDO |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2015-03-11
Ligands: 2VC, EDO
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Matrix Metalloproteinase-13 Complexed With Selective Inhibitor Compound Q1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2014-12-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, FMT, 1UA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: ZN, CA, FMT, 1UA, GOL
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Binding Mode, Selectivity And Potency Of N-Indolyl-Oxopyridinyl-4- Amino-Propanyl-Based Inhibitors Targeting Trypanosoma Cruzi Cyp51
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2014-11-26 Classification: OXIDOREDUCTASE Ligands: HEM, J5Y, SO4 |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: HEM, J5Y, SO4
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Crystal Structure Analysis Of Cruzain Bound To Vinyl Sulfone Analog Of Wrr-483 (Wrr-666)
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2014-11-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 2V5 |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-11-12
Ligands: 2V5
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Crystal Structure Of Trypanosoma Cruzi Cyp51 Bound To The Inhibitor (R)-N-(3-(1H-Indol-3-Yl)-1-Oxo-1-(Pyridin-4-Ylamino)Propan-2-Yl)-2-Fluoro-4-(4-(4-(Trifluoromethyl)Phenyl)Piperazin-1-Yl)Benzamide
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2014-09-03 Classification: OXIDOREDUCTASE Ligands: HEM, 26N, EDO, CL |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: HEM, 26N, EDO, CL
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Crystal Structure Of Trypanosoma Cruzi Cyp51 Bound To The Inhibitor (R)-N-(3-(1H-Indol-3-Yl)-1-Oxo-1-(Pyridin-4-Ylamino)Propan-2-Yl)-4-(4-(4-Chlorophenyl)Piperazin-1-Yl)-2-Fluorobenzamide.
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2014-09-03 Classification: OXIDOREDUCTASE Ligands: HEM, TW5, EDO, CL |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: HEM, TW5, EDO, CL
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Crystal Structure Of Trypanosoma Cruzi Cyp51 Bound To The Inhibitor (R)-N-(3-(1H-Indol-3-Yl)-1-Oxo-1-(Pyridin-4-Ylamino)Propan-2-Yl)-4-(4-(2,4-Difluorophenyl)Piperazin-1-Yl)-2-Fluorobenzamide.
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2014-08-20 Classification: OXIDOREDUCTASE Ligands: HEM, WVH, SO4, GOL |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2014-08-20
Ligands: HEM, WVH, SO4, GOL