Search Count: 52
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Crystal Structure Of Bcl-Xl In Complex With A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2024-10-16 Classification: APOPTOSIS Ligands: A1AFG, CD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: A1AFG, CD
 |
Crystal Structure Of Bcl-2 In Complex With Prodrug Abbv-167
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2021-04-14 Classification: APOPTOSIS Ligands: XZD |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: XZD
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Brd2_Bromodomain1 Complex With Inhibitor 744
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2020-01-29 Classification: SIGNALING PROTEIN Ligands: EDO, HWV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-29
Ligands: EDO, HWV
 |
Brd2_Bromodomain2 Complex With Inhibitor 744
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: HWV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: HWV
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Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-10-04 Classification: signaling protein/inhibitor Ligands: CJY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: CJY
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Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-10-04 Classification: signaling protein/inhibitor Ligands: CN7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: CN7
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The Novel P300/Cbp Inhibitor A-485 Uncovers A Unique Mechanism Of Action To Target Ar In Castrate Resistant Prostate Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-09-27 Classification: transferase/transferase INHIBITOR Ligands: 6TF, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: 6TF, NA
 |
Crystal Structure Of Human Nampt With A-1293201
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2017-06-28 Classification: Transferase/Transferase Inhibitor Ligands: 7T7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 7T7, SO4
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Crystal Structure Of Human Nampt With A-1326133
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2017-06-28 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 7TA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: SO4, 7TA
 |
Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2017-05-03 Classification: signaling protein/inhibitor Ligands: 9EA, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-03
Ligands: 9EA, ZN
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Discovery Of A Potent And Selective Bcl-Xl Inhibitor That Demonstrates Thrombocytopenia And Inhibits Tumor Growth In Vivo
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-07-22 Classification: APOPTOSIS/INHIBITOR Ligands: 3CQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-22
Ligands: 3CQ
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Bcl_2-Navitoclax Analog (With Indole) Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2014-01-29 Classification: APOPTOSIS REGULATOR/INHIBITOR Ligands: 1Y1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-29
Ligands: 1Y1
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Bcl_2-Navitoclax (Abt-263) Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-08-14 Classification: APOPTOSIS REGULATOR/INHIBITOR Ligands: 1XJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: 1XJ
 |
Bcl_2-Navitoclax Analog (Without Thiophenyl) Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-08-14 Classification: APOPTOSIS REGULATOR/INHIBITOR Ligands: 1XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: 1XV
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Crystal Structure Of Hsp90 With N-Aryl-Benzimidazolone I
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-09-21 Classification: CHAPERONE Ligands: MEX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-21
Ligands: MEX
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Crystal Structure Of Hsp90 With Ver-49009
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2011-09-21 Classification: CHAPERONE Ligands: BSM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-21
Ligands: BSM
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Crystal Structure Of Hsp90 With N-Aryl-Benzimidazolone Ii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2011-09-21 Classification: CHAPERONE Ligands: MEY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-21
Ligands: MEY
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Structure Of H-Chk1 Complexed With A767085
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: 76A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: 76A
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Structure Of H-Chk1 Complexed With Aa582939
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: A58 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: A58
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Structure Of H-Chk1 Complexed With A771129
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: 77A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: 77A