Search Count: 40
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Crystal Structure Of Egfr Exon20 Insertion Mutant In Complex With Enozertinib (Oric-114)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2025-11-12 Classification: SIGNALING PROTEIN Ligands: A1L8T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: A1L8T
 |
G-925 Bound To The Smarca4 (Brg1) Bromodomain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2022-08-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GGU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: GGU
 |
G-059 Bound To The Smarca4 (Brg1) Bromodomain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2022-08-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GJN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: GJN
 |
Structure Of The Human Jak1 Kinase Domain With Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KEJ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KEJ, GOL
 |
Structure Of The Human Jak1 Kinase Domain With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KEP, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KEP, GOL
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Structure Of The Human Jak1 Kinase Domain With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KES, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KES, GOL
 |
Structure Of The Human Jak1 Kinase Domain With Compound 39
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: GOL, KEV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: GOL, KEV
 |
Structure Of The Human Jak1 Kinase Domain With Compound 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KEY, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KEY, GOL
 |
Structure Of The Human Jak1 Kinase Domain With Compound 56
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KF1, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KF1, GOL
 |
Structure Of The Human Jak1 Kinase Domain With Compound 54
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KF4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KF4, GOL
 |
Taf1-Bd2 In Complex With Cpd27 (6-(But-3-En-1-Yl)-4-(1-Methyl-6-(Morpholine-4-Carbonyl)-1H-Benzo[D]Imidazol-4-Yl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-11-14 Classification: Transcription/Inhibitor Ligands: G9V |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: G9V
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Taf1-Bd2 In Complex With Cpd8 (6-(But-3-En-1-Yl)-4-(3-(Morpholine-4-Carbonyl)Phenyl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2018-10-31 Classification: Transcription/Inhibitor Ligands: G9Y |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: G9Y
 |
Crebbp Bromodomain In Complex With Cpd 4 (1-(1-(Cyclopropylmethyl)-3-(1H-Indol-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2018-08-08 Classification: PROTEIN BINDING/INHIBITOR Ligands: DMS, EDO, BKD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: DMS, EDO, BKD
 |
Crebbp Bromodomain In Complex With Cpd3 ((S)-1-(3-(6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9U7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9U7
 |
Crebbp Bromodomain In Complex With Cpd8 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2018-03-07 Classification: TRANSFERASE/INHIBITOR Ligands: 9UA, DMS, GOL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UA, DMS, GOL
 |
Crebbp Bromodomain In Complex With Cpd10 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9UD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UD
 |
Crebbp Bromodomain In Complex With Cpd17 (N,2,7-Trimethyl-2,3-Dihydro-4H-Benzo[B][1,4]Oxazine-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: SO4, 9UG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: SO4, 9UG
 |
Crebbp Bromodomain In Complex With Cpd19 (3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-N-Methyl-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridine-5-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2018-02-21 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9U4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: 9U4
 |
Crebbp Bromodomain In Complex With Cpd6 (Methyl 1H-Indole-3-Carboxylate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: DMS, C2Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: DMS, C2Y
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Crebbp Bromodomain In Complex With Cpd16 (5-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-N-Methyl-1H-Indole-3-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: C3J, EDO, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: C3J, EDO, NA