Search Count: 13
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: SAH, ZN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: SAH, ZN, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, X52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, X52
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3685032A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, UXM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, UXM
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Crystal Structure Of Gsk6157 Bound To Perk (R587-R1092, Delete A660-T867) At 2.34A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2014-09-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 27D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 27D
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Crystal Structure Of Gsk6414 Bound To Perk (R587-R1092, Delete A660-T867) At 2.28 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 0WH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: GOL, 0WH
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Crystal Structure Of Gsk6924 Bound To Perk (R587-R1092, Delete A660-T867) At 2.70 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 924 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: 924
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-(3-Amino-1H-Indazol-6-Yl)-N4-Ethyl-2,4-Pyrimidinediamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q0
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-[2-Amino-6-(4-Morpholinyl)-4-Pyrimidinyl]-1H-Indazol-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q1
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-{2-Amino-6-[(3R)-3-Methyl-4-Morpholinyl]-4-Pyrimidinyl}-1H-Indazol-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q2
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 4-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-N-Phenyl-2-Morpholinecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q3
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With (2R,5S)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-6-Methyl-N-Phenyl-3-Piperidinecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q4
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 1,1-Dimethylethyl {(3R,6S)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-6-Methyl-3-Piperidinyl}Carbamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Q5, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: 3Q5, SO4, GOL
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 1,1-Dimethylethyl{(3R,5R)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-5-Methyl-3-Piperidinyl}Carbamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Q6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: 3Q6, SO4