Search Count: 12
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Crystal Structure Of Human Lysophosphatidic Acid Receptor 1 In Complex With Ono9780307
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2015-06-03 Classification: TRANSPORT PROTEIN/inhibitor Ligands: ON7, 1WV |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: ON7, 1WV
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Crystal Structure Of Human Lysophosphatidic Acid Receptor 1 In Complex With Ono-9910539
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-06-03 Classification: TRANSPORT PROTEIN/inhibitor Ligands: ON9, 1WV |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: ON9, 1WV
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Crystal Structure Of Human Lysophosphatidic Acid Receptor 1 In Complex With Ono-3080573
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-06-03 Classification: TRANSPORT PROTEIN/inhibitor Ligands: ON3, 1WV |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: ON3, 1WV
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Quinazolines With Intra-Molecular Hydrogen Bonding Scaffold (Imhbs) As Pi3K/Mtor Dual Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2011-02-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3RE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-09
Ligands: 3RE
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Quinazolines With Intra-Molecular Hydrogen Bonding Scaffold (Imhbs) As Pi3K/Mtor Dual Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-02-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3RZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-09
Ligands: 3RZ
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Quinazolines With Intra-Molecular Hydrogen Bonding Scaffold (Imhbs) As Pi3K/Mtor Dual Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-02-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3PS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-09
Ligands: 3PS
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4-Methylpteridineones As Orally Active And Selective Pi3K/Mtor Dual Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2010-09-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OAW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-22
Ligands: OAW
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Hsp90 N-Terminal Domain In Complex With 4-Chloro-6-{[(2R)-2-(2-Methylphenyl)Pyrrolidin-1-Yl]Carbonyl}Benzene-1,3-Diol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2010-02-09 Classification: CHAPERONE Ligands: 4CD, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-09
Ligands: 4CD, DMS
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Hsp90 N-Terminal Domain In Complex With (1R)-2-(5-Chloro-2,4-Dihydroxybenzoyl)-N-Ethylisoindoline-1-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2010-02-09 Classification: CHAPERONE Ligands: 1RC, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-09
Ligands: 1RC, PO4
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Hsp90 N-Terminal Domain In Complex With 4-(1,3-Dihydro-2H-Isoindol-2-Ylcarbonyl)Benzene-1,3-Diol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-02-09 Classification: CHAPERONE Ligands: PFT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-09
Ligands: PFT
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Dihydroxylphenyl Amides As Inhibitors Of The Hsp90 Molecular Chaperone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2008-11-25 Classification: CHAPERONE Ligands: PYU, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-25
Ligands: PYU, PO4
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Dihydroxylphenyl Amides As Inhibitors Of The Hsp90 Molecular Chaperone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-11-25 Classification: CHAPERONE Ligands: PY9, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-25
Ligands: PY9, PO4
