Search Count: 9
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P110Delta/P85Alpha With Taselisib (Gdc-0032)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2017-01-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 799 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 799
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Imidazobenzoxepin Compound 3
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: SO4, 76Z |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: SO4, 76Z
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Benzoxepin Compound 2
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: 774, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 774, SO4
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Aryl Pyrrole Fragment 17
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: SO4, 76Y |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: SO4, 76Y
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Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 7KC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 7KC
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Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OL
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Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OL
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Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OQ
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Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OO
