Search Count: 9
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Crystal Structure Of Wild Type Egfr In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2022-12-07 Classification: HYDROLASE Ligands: R28 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: R28
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Crystal Structure Of Egfr_D770_N771Insnpg/V948R In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-12-07 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: R28, EDO, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: R28, EDO, CIT
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Structure Of Egfr_D770_N771Insnpg/V948R In Complex With Covalent Inhibitor Osimertinib.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2021-09-22 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: Q6K, EDO, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: Q6K, EDO, CIT
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Crystal Structure Of Anaplastic Lymphoma Kinase (Alk) Bound By Brigatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2018-12-12 Classification: TRANSFERASE Ligands: 6GY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-12
Ligands: 6GY
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Crystal Structure Of Kit In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-10-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0LI, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 0LI, PO4
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Crystal Structure Of Abl Kinase Domain Bound With A Dfg-Out Inhibitor Ap24534
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-12-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0LI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-12-15
Ligands: 0LI
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Crystal Structure Of Abl T315I Mutant Kinase Domain Bound With A Dfg-Out Inhibitor Ap24589
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2010-12-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: XY3 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-12-15
Ligands: XY3
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Ap24534, A Pan-Bcr-Abl Inhibitor For Chronic Myeloid Leukemia, Potently Inhibits The T315I Mutant And Overcomes Mutation-Based Resistance
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-11-03 Classification: TRANSFERASE Ligands: 0LI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2009-11-03
Ligands: 0LI
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Fk506 Binding Protein Mutant, Homodimeric Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2000-08-09 Classification: ISOMERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2000-08-09
