Search Count: 22
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Cdk9/Cyclin T1 In Complex With Kb-0742
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.75 Å Release Date: 2023-12-06 Classification: TRANSCRIPTION Ligands: VQE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: VQE
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Type 1 Prmt In Complex With The Inhibitor Gsk3368715
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2019-07-10 Classification: ANTITUMOR PROTEIN Ligands: SAH, KZS, GOL, DTT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: SAH, KZS, GOL, DTT
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Crystal Structure Of Smyd2 With Sam And Epz033294
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-04-25 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SAM, ZN, 8WG, PEG, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-25
Ligands: SAM, ZN, 8WG, PEG, EDO, GOL
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Estrogen Receptor Alpha Y537S Covalently Bound To Antagonist H3B-5942.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2018-03-21 Classification: nuclear protein/antagonist Ligands: F3D, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: F3D, EDO, DMS
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Estrogen Receptor Alpha Y537S Bound To Antagonist H3B-9224.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2018-03-21 Classification: nuclear protein/antagonist Ligands: F3D, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: F3D, EDO
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Crystal Structure Of Smyd3 With Sam And Epz028862
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2018-03-07 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: ZN, SAM, 8WD, PEG, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: ZN, SAM, 8WD, PEG, DMS, EDO
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Crystal Structure Of Carm1 With Epz022302 And Sah
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2018-02-07 Classification: TRANSFERASE Ligands: SAH, BW4, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-07
Ligands: SAH, BW4, GOL, SO4
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Crystal Structure Of Carm1 With Compound 2 And Sah
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-02-07 Classification: TRANSFERASE Ligands: SAH, BW7, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-07
Ligands: SAH, BW7, GOL
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Crystal Structure Of Fgfr1-Y563C (Fgfr4 Surrogate) Covalently Bound To H3B-6527
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-05-24 Classification: transferase/transferase inhibitor Ligands: 9ES, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 9ES, SO4, EDO
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Crystal Structure Of Prmt5:Mep50 With Compound 8 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 5QJ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SFG, 5QJ, GOL
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Crystal Structure Of Prmt5:Mep50 With Compound 9 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 5QH, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SFG, 5QH, GOL
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Crystal Structure Of Prmt5:Mep50 With Compound 10 And Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 5QK, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SAM, 5QK, GOL
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Crystal Structure Of Prmt5:Mep50 With Compound 15 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 5QL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SFG, 5QL, GOL
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Crystal Structure Of Smyd3 With Sam And Oxindole Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2015-09-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, SAM, 4ZW, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-09
Ligands: ZN, SAM, 4ZW, EDO
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Crystal Structure Of Smyd3 With Sam And Epz030456
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-09-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, SAM, 4ZX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-09
Ligands: ZN, SAM, 4ZX
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 3XV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SFG, 3XV, GOL
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 3XV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAM, 3XV, GOL
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sah
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAH, 3XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAH, 3XV
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Crystal Structure Of Human Protein Arginine Methyltransferase Prmt6 Bound To Sah And An Aryl Pyrazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: SAH, 49K, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAH, 49K, GOL
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Crystal Structure Of Human Protein Arginine Methyltransferase Prmt6 Bound To Sah And Epz020411
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: SAH, 49L, MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAH, 49L, MG, GOL
