Search Count: 70
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Crystal Structure Of Sars Cov-2 3Cl Protease In Complex With Gsk4365096A
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2024-03-13 Classification: HYDROLASE Ligands: WTE |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-03-13
Ligands: WTE
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Crystal Structure Of Sars Cov-2 3Cl Protease In Complex With Gsk4365097A
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2024-02-14 Classification: HYDROLASE Ligands: WTV, GOL, CL |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: WTV, GOL, CL
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Crystal Structure Of Sars Cov-2 3Cl Protease In Complex With Gsk4365096A
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2024-02-14 Classification: HYDROLASE Ligands: A1ADS |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: A1ADS
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Sara Cov-2 3C-Like Protease In Complex With Gsk3487016A
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-02-14 Classification: HYDROLASE Ligands: WYR, EDO |
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: WYR, EDO
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X-Ray Structure Of Furin Bound To Bos-318, A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2022-01-12 Classification: HYDROLASE/INHIBITOR Ligands: CA, XTA, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: CA, XTA, EDO
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Hpgds Complexed With An Aza-Quinoline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-11-04 Classification: HYDROLASE Ligands: GSH, SWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-04
Ligands: GSH, SWS
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H-Pgds Complexed With Inhibitor 1Y
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2020-11-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GSH, EDO, TJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-04
Ligands: GSH, EDO, TJG
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Crystal Structure Of Rip1 Kinase In Complex With Gsk3145095
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2019-07-03 Classification: TRANSFERASE Ligands: K8K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-03
Ligands: K8K
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Hpgds Complexed With A Quinoline-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: GSH, KCD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-27
Ligands: GSH, KCD
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Rat Hpgds Complexed With A Quinoline
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: GSH, KDV |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2019-03-27
Ligands: GSH, KDV
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Bmp1 Complexed With A Reverse Hydroxymate - Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-08-08 Classification: HYDROLASE Ligands: SCN, ZN, EVV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SCN, ZN, EVV, EDO
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Bmp1 Complexed With A Reverse Hydroxamate - Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2018-08-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, E7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: ZN, E7D
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Bmp1 Complexed With A Reverse Hydroxymate - Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-08-08 Classification: HYDROLASE Ligands: EDO, ZN, E8M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: EDO, ZN, E8M
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Bmp1 Complexed With (2~{S})-2-[[(1~{R},3~{S},4~{S})-2-[(2~{R})-2-[2-(Oxidanylamino)-2-Oxidanylidene-Ethyl]Heptanoyl]-2-Azabicyclo[2.2.1]Heptan-3-Yl]Carbonylamino]-2-Phenyl-Ethanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-08-08 Classification: HYDROLASE Ligands: SCN, ZN, E8P, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SCN, ZN, E8P, EDO
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Bmp1 Complexed With A Hydroxamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2018-08-08 Classification: HYDROLASE Ligands: SCN, ZN, E8J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SCN, ZN, E8J
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Bmp1 Complexed With A Hydroxamate - Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2018-08-08 Classification: HYDROLASE Ligands: SCN, ZN, E8S, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SCN, ZN, E8S, EDO
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Rip1 Kinase ( Flag 1-294, C34A, C127A, C233A, C240A) With Gsk772
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2017-07-05 Classification: transferase/transferase inhibitor Ligands: 7MJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-05
Ligands: 7MJ
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Factor Viia In Complex With The Inhibitor 3-{[(2R)-17-Ethyl-4-Methyl-3,12-Dioxo-7-[(Propan-2-Yl)Sulfonyl]-13-Oxa-4,11-Diazatricyclo[14.2.2.1~6,10~]Henicosa-1(18),6(21),7,9,16,19-Hexaen-2-Yl]Amino}Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-05-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 82J, CA, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 82J, CA, SO4, GOL
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Factor Viia In Complex With The Inhibitor (5R)-5-[(1-Aminoisoquinolin-6-Yl)Amino]-19-(Cyclopropylsulfonyl)-3-Methyl-13-Oxa-3,15-Diazatricyclo[14.3.1.1~6,10~]Henicosa-1(20),6(21),7,9,16,18-Hexaene-4,14-Dione
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-02-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 7KQ, CA, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-01
Ligands: 7KQ, CA, SO4, GOL
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Factor Viia In Complex With The Inhibitor (11R)-11-[(1-Aminoisoquinolin-6-Yl)Amino]-16-(Cyclopropylsulfonyl)-13-Methyl-2,13-Diazatricyclo[13.3.1.1~6,10~]Icosa-1(19),6(20),7,9,15,17-Hexaene-3,12-Dione
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2017-02-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 7KR, CA, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-01
Ligands: 7KR, CA, SO4, GOL
