Search Count: 17
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Structure Of Human Beta 1,3-N-Acetylglucosaminyltransferase 2 With Compound 7J
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2023-12-06 Classification: TRANSFERASE Ligands: X18, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: X18, EDO
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Structure Of Human Beta 1,3-N-Acetylglucosaminyltransferase 2 With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2023-12-06 Classification: TRANSFERASE Ligands: NAG, FKX, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: NAG, FKX, GOL, CL
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Structure Of Human Beta 1,3-N-Acetylglucosaminyltransferase 2 With Compound 8A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-12-06 Classification: TRANSFERASE Ligands: MN, HI8, NAG, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: MN, HI8, NAG, PEG
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Crystal Structure Of Human Kras G12C Covalently Bound To A Phthalazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, OJ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: MG, GDP, OJ1
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Crystal Structure Of Human Kras G12C Covalently Bound To A Quinazolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: GDP, CA, OHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: GDP, CA, OHY
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolodihydropyrrolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: JYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: JYG, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolopyrrolone Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-06-22 Classification: transferase/transferase inhibitor Ligands: 6CD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 6CD, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Macrocyclic Quinoxaline-Pyrrolodihydropiperidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-04 Classification: transferase/transferase inhibitor Ligands: 5QO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 5QO, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiazolamine-Indazole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U5, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiadiazolamine-Indole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U6, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U6, GOL
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Co-Crystal Structure Of Pim1 With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3UR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 3UR
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Crystal Structure Of Human Pim-1 Kinase In Complex With An Aminooxadiazole-Indole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 38W, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 38W, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With An Azaspiro Pyrazinyl-Indazole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-02-04 Classification: transferase/transferase inhibitor Ligands: GOL, 3U1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: GOL, 3U1
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Crystal Structure Of Human Pi3K-Gamma In Complex With Amg511
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2012-08-29 Classification: Transferase/Inhibitor Ligands: SO4, 14K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: SO4, 14K
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Crystal Structure Of Human Pi3K-Gamma In Complex With A Pyridyl-Triazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2012-05-16 Classification: Transferase/Inhibitor Ligands: SO4, 0KO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: SO4, 0KO
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P38 Complexed With A Quinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2008-10-14 Classification: TRANSFERASE Ligands: P40 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-14
Ligands: P40
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P38 Complex With A Phthalazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2008-10-07 Classification: TRANSFERASE Ligands: A17 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: A17
